SCHEMBL2369708

SCHEMBL2369708

CNC(=O)c1c(-c2ccc(F)cc2)oc2cc(NC(C)=O)c(-c3cccc(C(=O)N(c4ccccc4)C4CC4)c3)cc12

nearest known ligand 0.50

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.43
CYP2C8 P10632 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1918986 0.90 CYP3A4 (0.41) CYP3A4CYP2C8
SCHEMBL1919554 0.89 CYP3A4 (0.45) CYP3A4CYP2C8
SCHEMBL1919876 0.87 CYP3A4 (0.50) CYP3A4CYP2C8
SCHEMBL1920422 0.86 CYP3A4 (0.43) CYP3A4CYP2C8
SCHEMBL1918583 0.86 CYP3A4 (0.39) CYP3A4CYP2C8
SCHEMBL1918510 0.84 CYP3A4 (0.49) CYP3A4CYP2C8
SCHEMBL1918518 0.83 CYP3A4 (0.41) CYP3A4
SCHEMBL1919024 0.82 CYP2C8 (0.56) CYP3A4CYP2C8
SCHEMBL1918584 0.82 CYP3A4 (0.47) CYP3A4
SCHEMBL1918465 0.81 CYP2C8 (0.55) CYP3A4CYP2C8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2545042-A1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C Bristol-Myers Squibb Company (US) 2013-01-16 EP disclosed
WO-2011112191-A1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C BRISTOL-MYERS SQUIBB COMPANY (US) 2011-09-15 WO disclosed