SCHEMBL2369796

SCHEMBL2369796

Nc1ccc2nc(Nc3cccc(NC4CCC(O)CC4)n3)sc2c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITK Q08881 13/20 0.54
LCK P06239 14/20 0.50
AURKB Q96GD4 12/20 0.50
EGFR P00533 1/20 0.49
INSR P06213 1/20 0.49
SRC P12931 1/20 0.49
TEC P42680 1/20 0.49
TXK P42681 1/20 0.49
BMX P51813 1/20 0.49
BTK Q06187 1/20 0.49
LRRK2 Q5S007 1/20 0.49
CAMKK2 Q96RR4 1/20 0.49
IRAK4 Q9NWZ3 1/20 0.49
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
MEN1 O00255 1/20 0.47
GFER P55789 1/20 0.47
KMT2A Q03164 1/20 0.47
CCNT1 O60563 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2369789 1.00 ITK (0.54) ITKLCKAURKBEGFRINSR
SCHEMBL2370452 0.87 LCK (0.64) ITKLCKAURKBEGFRINSR
SCHEMBL2370446 0.87 LCK (0.64) ITKLCKAURKBEGFRINSR
SCHEMBL2369954 0.87 ITK (0.54) ITKLCKAURKBEGFRINSR
SCHEMBL2369949 0.87 ITK (0.54) ITKLCKAURKBEGFRINSR
SCHEMBL2382012 0.85 ITK (0.67) ITKLCKAURKBEGFRINSR
SCHEMBL2382006 0.85 ITK (0.67) ITKLCKAURKBEGFRINSR
SCHEMBL2396679 0.85 ITK (0.57) ITKLCKAURKBEGFRINSR
SCHEMBL2396683 0.85 ITK (0.57) ITKLCKAURKBEGFRINSR
SCHEMBL2397647 0.84 ABL1 (0.56) ITKLCKAURKBEGFRINSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011110575-A1 DERIVATIVES OF 2-[2-(BENZO- OR PYRIDO-) THIAZOLYLAMINO]-6-AMINOPYRIDINE, USEFUL IN THE TREATMENT OF RESPIRATORIC, ALLERGIC OR INFLAMMATORY DISEASES GLAXO GROUP LIMITED (GB) 2011-09-15 WO disclosed