SCHEMBL2397647

SCHEMBL2397647

Nc1ccc(-c2ccc3nc(Nc4cccc(N[C@H]5CC[C@H](O)CC5)n4)sc3c2)cn1

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 2/20 0.56
PIK3CA P42336 4/20 0.51
CYP3A4 P08684 1/20 0.51
ITK Q08881 10/20 0.48
AURKB Q96GD4 9/20 0.45
LCK P06239 8/20 0.45
IRAK4 Q9NWZ3 2/20 0.44
EGFR P00533 1/20 0.44
INSR P06213 1/20 0.44
SRC P12931 1/20 0.44
TEC P42680 1/20 0.44
TXK P42681 1/20 0.44
BMX P51813 1/20 0.44
BTK Q06187 1/20 0.44
LRRK2 Q5S007 1/20 0.44
CAMKK2 Q96RR4 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2397651 1.00 ABL1 (0.56) ABL1PIK3CACYP3A4ITKAURKB
SCHEMBL2397008 0.86 ITK (0.48) ABL1ITKAURKBLCKIRAK4
SCHEMBL2396998 0.86 ITK (0.48) ABL1ITKAURKBLCKIRAK4
SCHEMBL2401516 0.86 PIK3CG (0.54) PIK3CAITKAURKBLCKIRAK4
SCHEMBL2401498 0.86 PIK3CG (0.54) PIK3CAITKAURKBLCKIRAK4
SCHEMBL2396683 0.86 ITK (0.57) ABL1ITKAURKBLCKIRAK4
SCHEMBL2396679 0.86 ITK (0.57) ABL1ITKAURKBLCKIRAK4
SCHEMBL2369714 0.86 PIK3CA (0.52) ABL1PIK3CAITKAURKBLCK
SCHEMBL2369722 0.86 PIK3CA (0.52) ABL1PIK3CAITKAURKBLCK
SCHEMBL2370102 0.85 ITK (0.51) ABL1PIK3CAITKAURKBLCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011110575-A1 DERIVATIVES OF 2-[2-(BENZO- OR PYRIDO-) THIAZOLYLAMINO]-6-AMINOPYRIDINE, USEFUL IN THE TREATMENT OF RESPIRATORIC, ALLERGIC OR INFLAMMATORY DISEASES GLAXO GROUP LIMITED (GB) 2011-09-15 WO disclosed