SCHEMBL2370058

SCHEMBL2370058

CC(C)(C)NC(=O)c1cncc(B(O)O)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 1/20 0.41
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C19 P33261 1/20 0.39
POLB P06746 3/20 0.38
MAPT P10636 1/20 0.38
KDM4E B2RXH2 1/20 0.36
PTGS2 P35354 2/20 0.36
PTGS1 P23219 1/20 0.36
PRKAB2 O43741 1/20 0.35
PRKAG1 P54619 1/20 0.35
PRKAA2 P54646 1/20 0.35
PRKAA1 Q13131 1/20 0.35
PRKAG3 Q9UGI9 1/20 0.35
PRKAG2 Q9UGJ0 1/20 0.35
PRKAB1 Q9Y478 1/20 0.35
TRPV1 Q8NER1 2/20 0.35
IRAK4 Q9NWZ3 1/20 0.35
HPGD P15428 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23243007 0.81 RAF1 (0.44) HPGDSKDM4EPTGS2PTGS1
SCHEMBL2735676 0.78 HCAR2 (0.56) HPGDS
SCHEMBL13701655 0.77 ABL1 (0.50) HPGDSCYP1A2CYP3A4CYP2C19IRAK4
SCHEMBL10288898 0.77 KDM4E (0.62) CYP1A2CYP3A4CYP2C19POLBKDM4E
SCHEMBL5105519 0.75 MKNK1 (0.45) CYP1A2CYP3A4POLBKDM4E
SCHEMBL520859 0.75 LMNA (0.49) CYP2C19
SCHEMBL961277 0.75 ATM (0.61) CYP2C19POLBKDM4E
SCHEMBL1501699 0.74 ATM (0.40) CYP1A2CYP3A4CYP2C19SMN1; SMN2
SCHEMBL1961940 0.74 TRPV1 (0.58) MAPTTRPV1
Hydrochloric Acid SCHEMBL1054647 0.73 ATM (0.59) CYP2C19POLBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed
WO-2014106800-A2 SUBSTITUTED 2-AMINO PYRIMIDINE DERIVATIVES AS KINASE INHIBITORS AURIGENE DISCOVERY TECHNOLOGIES LIMITED (IN) 2014-07-10 WO disclosed
WO-2012174312-A2 BENZIMIDAZOLE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-12-20 WO disclosed
WO-2012087938-A1 QUINAZOLINONE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-06-28 WO disclosed
WO-2011110575-A1 DERIVATIVES OF 2-[2-(BENZO- OR PYRIDO-) THIAZOLYLAMINO]-6-AMINOPYRIDINE, USEFUL IN THE TREATMENT OF RESPIRATORIC, ALLERGIC OR INFLAMMATORY DISEASES GLAXO GROUP LIMITED (GB) 2011-09-15 WO disclosed