SCHEMBL2370604

SCHEMBL2370604

OC1CCC(Nc2cccc(Nc3nc4ccc(-c5ccoc5)cc4s3)n2)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITK Q08881 11/20 0.49
AURKB Q96GD4 10/20 0.45
LCK P06239 9/20 0.45
EGFR P00533 1/20 0.44
INSR P06213 1/20 0.44
SRC P12931 1/20 0.44
TEC P42680 1/20 0.44
TXK P42681 1/20 0.44
BMX P51813 1/20 0.44
BTK Q06187 1/20 0.44
LRRK2 Q5S007 1/20 0.44
CAMKK2 Q96RR4 1/20 0.44
IRAK4 Q9NWZ3 1/20 0.44
USP2 O75604 3/20 0.41
ALDH1A1 P00352 3/20 0.41
CYP1A2 P05177 3/20 0.41
CYP2D6 P10635 3/20 0.41
HSD17B10 Q99714 3/20 0.41
MEN1 O00255 2/20 0.41
CYP3A4 P08684 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2370596 1.00 ITK (0.49) ITKAURKBLCKEGFRINSR
SCHEMBL2396683 0.87 ITK (0.57) ITKAURKBLCKEGFRINSR
SCHEMBL2396679 0.87 ITK (0.57) ITKAURKBLCKEGFRINSR
SCHEMBL2398141 0.86 ITK (0.48) ITKAURKBLCKEGFRINSR
SCHEMBL2398154 0.86 ITK (0.48) ITKAURKBLCKEGFRINSR
SCHEMBL2370102 0.85 ITK (0.51) ITKAURKBLCKEGFRINSR
SCHEMBL2370095 0.85 ITK (0.51) ITKAURKBLCKEGFRINSR
SCHEMBL2396030 0.83 ITK (0.49) ITKAURKBLCKEGFRINSR
SCHEMBL2369714 0.83 PIK3CA (0.52) ITKAURKBLCKEGFRINSR
SCHEMBL2396032 0.83 ITK (0.49) ITKAURKBLCKEGFRINSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011110575-A1 DERIVATIVES OF 2-[2-(BENZO- OR PYRIDO-) THIAZOLYLAMINO]-6-AMINOPYRIDINE, USEFUL IN THE TREATMENT OF RESPIRATORIC, ALLERGIC OR INFLAMMATORY DISEASES GLAXO GROUP LIMITED (GB) 2011-09-15 WO disclosed