SCHEMBL2370682

SCHEMBL2370682

COc1ccc2c(c1)CN(C1CCCC1)CC2

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 7/20 0.53
CYP2D6 P10635 3/20 0.52
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
ATM Q13315 1/20 0.52
DRD1 P21728 4/20 0.51
DRD5 P21918 3/20 0.51
DRD2 P14416 3/20 0.51
DRD3 P35462 2/20 0.51
DRD4 P21917 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16855300 0.87 HRH3 (0.56) HRH3CYP2D6DRD1DRD5DRD2
Hydrochloric Acid SCHEMBL16824558 0.86 HRH3 (0.55) HRH3CYP2D6DRD1DRD5DRD2
SCHEMBL18186150 0.83 ADRA1A (0.52) HRH3MEN1KMT2AATMDRD1
SCHEMBL16846277 0.82 HRH3 (0.56) HRH3CYP2D6DRD1DRD5DRD2
SCHEMBL24039956 0.81 HIF1A (0.56) MEN1KMT2AATMDRD1DRD5
SCHEMBL11261438 0.81 DRD1 (0.49) HRH3DRD1DRD5DRD2DRD3
Hydrochloric Acid SCHEMBL16824528 0.81 HRH3 (0.55) HRH3CYP2D6DRD1DRD5DRD2
SCHEMBL15759170 0.80 HRH3 (0.43) HRH3CYP2D6
SCHEMBL20220387 0.78 CHRM2 (0.52) HRH3DRD1DRD2
SCHEMBL16855353 0.78 STS (0.53) HRH3MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011116356-A2 POSITIVE ALLOSTERIC MODULATORS OF GROUP II MGLURS SANFORD-BURNHAM MEDICAL RESEARCH INSTITUTE (US) 2011-09-22 WO disclosed