SCHEMBL2370728

SCHEMBL2370728

Fc1cc(Cc2ccccn2)cc(F)n1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.51
ASIC3 Q9UHC3 1/20 0.43
HRH3 Q9Y5N1 2/20 0.42
HRH1 P35367 1/20 0.41
HRH4 Q9H3N8 1/20 0.41
KDM4E B2RXH2 1/20 0.41
LMNA P02545 1/20 0.41
TAAR1 Q96RJ0 1/20 0.41
ALDH1A1 P00352 1/20 0.41
ALOX15 P16050 1/20 0.41
MAPT P10636 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
LIN28A Q9H9Z2 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
RAB9A P51151 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30063557 0.81 L3MBTL1 (0.51) L3MBTL1ASIC3HRH3HRH1HRH4
SCHEMBL3233668 0.77 L3MBTL1 (0.65) L3MBTL1HRH3HRH1HRH4KDM4E
SCHEMBL4212164 0.76 KDM4E (0.61) L3MBTL1KDM4ETAAR1ALDH1A1MAPT
SCHEMBL15081590 0.76 L3MBTL1 (0.58) L3MBTL1ASIC3HRH3HRH1HRH4
SCHEMBL64435 0.76 L3MBTL1 (0.68) L3MBTL1HRH3HRH1HRH4LMNA
SCHEMBL29373231 0.76 L3MBTL1 (0.68) L3MBTL1HRH3HRH1HRH4LMNA
SCHEMBL7083429 0.76 L3MBTL1 (0.53) L3MBTL1ASIC3HRH3HRH1HRH4
SCHEMBL30064008 0.75 L3MBTL1 (0.49) L3MBTL1HRH3HRH1HRH4ALDH1A1
SCHEMBL41191 0.75 L3MBTL1 (0.59) L3MBTL1ASIC3HRH3HRH1HRH4
SCHEMBL29830938 0.75 L3MBTL1 (0.59) L3MBTL1ASIC3HRH3HRH1HRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011110575-A1 DERIVATIVES OF 2-[2-(BENZO- OR PYRIDO-) THIAZOLYLAMINO]-6-AMINOPYRIDINE, USEFUL IN THE TREATMENT OF RESPIRATORIC, ALLERGIC OR INFLAMMATORY DISEASES GLAXO GROUP LIMITED (GB) 2011-09-15 WO disclosed
WO-2011110575-A1 DERIVATIVES OF 2-[2-(BENZO- OR PYRIDO-) THIAZOLYLAMINO]-6-AMINOPYRIDINE, USEFUL IN THE TREATMENT OF RESPIRATORIC, ALLERGIC OR INFLAMMATORY DISEASES GLAXO GROUP LIMITED (GB) 2011-09-15 WO disclosed