SCHEMBL23712415

SCHEMBL23712415

O=c1[nH]c(Nc2ccc(N3CCOCC3)cc2)ncc1Cl

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK10 P53779 3/20 0.50
MAPT P10636 3/20 0.49
TSHR P16473 1/20 0.49
NR4A1 P22736 1/20 0.49
EGFR P00533 1/20 0.48
ZAP70 P43403 2/20 0.47
CCNK O75909 1/20 0.47
CCNA2 P20248 1/20 0.47
CDK2 P24941 1/20 0.47
CCND3 P30281 1/20 0.47
CDK9 P50750 1/20 0.47
CDK6 Q00534 1/20 0.47
PKMYT1 Q99640 2/20 0.47
INSR P06213 1/20 0.47
IGF1R P08069 1/20 0.47
PTK2 Q05397 1/20 0.47
PTK2B Q14289 1/20 0.47
SLC2A1 P11166 1/20 0.46
MAPK8 P45983 1/20 0.46
MAPK9 P45984 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23704664 0.86 ALK (0.54) EGFRCCNKCCNA2CDK2CCND3
SCHEMBL16423097 0.78 MAPK10 (0.49) MAPK10MAPTCDK2SLC2A1MAPK8
SCHEMBL4075886 0.76 SYK (0.46) MAPK10MAPTZAP70CCND3MAPK8
SCHEMBL15349719 0.76 MAPT (0.62) MAPTPTK2BSLC2A1SYKALDH1A1
SCHEMBL994128 0.75 MEN1 (0.50) MAPTLRRK2ALDH1A1LMNAXBP1
SCHEMBL2061358 0.74 MAPT (0.62) MAPK10MAPTTSHRNR4A1EGFR
SCHEMBL4382248 0.73 TTBK1 (0.56) MAPTZAP70PTK2TP53MAPK1
SCHEMBL23704665 0.73 CCNK (0.65) MAPK10MAPTEGFRCCNKCCNA2
SCHEMBL23704673 0.72 PKMYT1 (0.69) MAPK10EGFRCCNKCCNA2CDK2
SCHEMBL14330684 0.72 EGFR (0.49) TSHREGFRZAP70CCNA2CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021155185-A1 AMINOPYRIMIDINYLAMINOBENZONITRILE DERIVATIVES AS NEK2 INHIBITORS SUMITOMO DAINIPPON PHARMA ONCOLOGY, INC. (US) 2021-08-05 WO disclosed