SCHEMBL2371305

SCHEMBL2371305

O=C(O)NC1=NC2(CS1)c1cc(-c3cccnc3F)ccc1Oc1cnc(Cl)cc12

nearest known ligand 0.49

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.49
CTSD P07339 10/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2372292 0.89 BACE1 (0.45) BACE1CTSD
SCHEMBL2371065 0.86 BACE1 (0.64) BACE1CTSD
SCHEMBL2370764 0.84 BACE1 (0.65) BACE1CTSD
SCHEMBL2522054 0.83 BACE1 (0.47) BACE1CTSD
SCHEMBL2522053 0.83 BACE1 (0.47) BACE1CTSD
SCHEMBL14629827 0.81 BACE1 (0.51) BACE1CTSD
SCHEMBL2517702 0.77 BACE1 (0.58) BACE1CTSD
SCHEMBL2517714 0.77 BACE1 (0.58) BACE1CTSD
SCHEMBL15418854 0.77 BACE1 (0.55) BACE1CTSD
SCHEMBL15418837 0.77 BACE1 (0.55) BACE1CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8883782-B2 Spiro-tetracyclic ring compounds as beta-secretase modulators and methods of use AMGEN INC. (US) 2014-11-11 US disclosed
EP-2547685-A1 SPIRO-TETRACYCLIC RING COMPOUNDS AS BETA - SECRETASE MODULATORS Amgen Inc. (US) 2013-01-23 EP disclosed
WO-2011115938-A1 SPIRO-TETRACYCLIC RING COMPOUNDS AS BETA - SECRETASE MODULATORS AMGEN INC. (US) 2011-09-22 WO disclosed