SCHEMBL2371326

SCHEMBL2371326

CC(C(=O)O)c1ncncc1F.[BaH2]

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 6/20 0.38
AKR1C2 P52895 6/20 0.38
CYP3A4 P08684 6/20 0.36
LMNA P02545 3/20 0.36
CYP2C9 P11712 2/20 0.34
CYP2C19 P33261 2/20 0.34
CYP2B6 P20813 1/20 0.34
CYP3A5 P20815 1/20 0.34
CYP3A7 P24462 1/20 0.34
MAPK1 P28482 1/20 0.34
CYP3A43 Q9HB55 1/20 0.34
CYP46A1 Q9Y6A2 1/20 0.34
PTGS1 P23219 3/20 0.33
PTGS2 P35354 3/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
FABP2 P12104 1/20 0.33
TSHR P16473 1/20 0.33
AKR1C4 P17516 1/20 0.33
ADRA2B P18089 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2370298 0.97 AKR1C3 (0.38) AKR1C3AKR1C2CYP3A4LMNACYP2C9
SCHEMBL2371309 0.81 CYP3A4 (0.36) CYP3A4LMNACYP2C9CYP2C19CYP2B6
Potassium Ion SCHEMBL2370572 0.81 CYP3A4 (0.36) CYP3A4LMNACYP2C9CYP2C19CYP2B6
Lithium Ion SCHEMBL2370296 0.81 CYP3A4 (0.36) CYP3A4LMNACYP2C9CYP2C19CYP2B6
SCHEMBL14562495 0.80 HCAR2 (0.34) AKR1C3AKR1C2CYP3A4LMNACYP2C9
SCHEMBL1553635 0.76 CYP3A4 (0.40) CYP3A4LMNACYP2C9CYP2C19CYP2B6
SCHEMBL2625489 0.75 CYP11B1 (0.40) CYP3A4LMNACYP2C9CYP2C19CYP2B6
SCHEMBL12298618 0.73 CYP3A4 (0.46) CYP3A4LMNACYP2C9CYP2C19CYP2B6
SCHEMBL5340414 0.72 CYP3A4 (0.37) CYP3A4LMNACYP2C9CYP2C19CYP2B6
SCHEMBL29009979 0.72 AKR1C3 (0.42) AKR1C3AKR1C2CYP3A4LMNACYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2545039-A1 A PROCESS FOR MAKING VORICONAZOLE Synthon BV (NL) 2013-01-16 EP disclosed
WO-2011110198-A1 A PROCESS FOR MAKING VORICONAZOLE SYNTHRON B.V. (NL) 2011-09-15 WO disclosed