SCHEMBL2371309

SCHEMBL2371309

CC(C(=O)[O-])c1ncncc1F.CC(C(=O)[O-])c1ncncc1F.[Ba+2]

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 6/20 0.36
CYP2C9 P11712 1/20 0.34
CYP2B6 P20813 1/20 0.34
CYP3A5 P20815 1/20 0.34
CYP3A7 P24462 1/20 0.34
MAPK1 P28482 1/20 0.34
CYP2C19 P33261 1/20 0.34
CYP3A43 Q9HB55 1/20 0.34
CYP46A1 Q9Y6A2 1/20 0.34
LMNA P02545 1/20 0.34
NLRP3 Q96P20 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2370533 0.97 CYP3A4 (0.36) CYP3A4CYP2C9CYP2B6CYP3A5CYP3A7
SCHEMBL2370196 0.97 CYP3A4 (0.36) CYP3A4CYP2C9CYP2B6CYP3A5CYP3A7
Potassium Ion SCHEMBL2370572 0.97 CYP3A4 (0.36) CYP3A4CYP2C9CYP2B6CYP3A5CYP3A7
Lithium Ion SCHEMBL2370296 0.97 CYP3A4 (0.36) CYP3A4CYP2C9CYP2B6CYP3A5CYP3A7
SCHEMBL2370540 0.85 TSHR (0.36) CYP3A4CYP2C9CYP2B6CYP3A5CYP3A7
SCHEMBL2371326 0.81 AKR1C3 (0.38) CYP3A4CYP2C9CYP2B6CYP3A5CYP3A7
SCHEMBL1553635 0.74 CYP3A4 (0.40) CYP3A4CYP2C9CYP2B6CYP3A5CYP3A7
SCHEMBL12298618 0.72 CYP3A4 (0.46) CYP3A4CYP2C9CYP2B6CYP3A5CYP3A7
SCHEMBL5340414 0.71 CYP3A4 (0.37) CYP3A4CYP2C9CYP2B6CYP3A5CYP3A7
SCHEMBL22368312 0.70 CYP3A4 (0.40) CYP3A4CYP2C9CYP2B6CYP3A5CYP3A7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2545039-A1 A PROCESS FOR MAKING VORICONAZOLE Synthon BV (NL) 2013-01-16 EP disclosed
WO-2011110198-A1 A PROCESS FOR MAKING VORICONAZOLE SYNTHRON B.V. (NL) 2011-09-15 WO disclosed