SCHEMBL23728162

SCHEMBL23728162

CC1CCN(Cc2ccc(NC(=O)NCc3ccc(Cl)cc3)cc2)C1=O

nearest known ligand 0.59

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 1/20 0.59
HTR2A P28223 1/20 0.59
MCHR1 Q99705 1/20 0.59
RAB9A P51151 3/20 0.57
NPC1 O15118 3/20 0.57
POLB P06746 1/20 0.54
LSS P48449 1/20 0.54
TP53 P04637 1/20 0.52
NAMPT P43490 3/20 0.51
ERCC1 P07992 1/20 0.49
ERCC4 Q92889 1/20 0.49
EPHX2 P34913 2/20 0.48
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
CNR1 P21554 1/20 0.46
HRH3 Q9Y5N1 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23728122 1.00 CHRM1 (0.59) CHRM1HTR2AMCHR1RAB9ANPC1
SCHEMBL23747508 1.00 CHRM1 (0.59) CHRM1HTR2AMCHR1RAB9ANPC1
SCHEMBL26102031 0.94 CHRM1 (0.57) CHRM1HTR2AMCHR1RAB9ANPC1
SCHEMBL26101652 0.94 CHRM1 (0.57) CHRM1HTR2AMCHR1RAB9ANPC1
SCHEMBL23747458 0.94 CHRM1 (0.57) CHRM1HTR2AMCHR1RAB9ANPC1
SCHEMBL23747337 0.88 SMN1; SMN2 (0.58) MCHR1RAB9ANPC1POLBNAMPT
SCHEMBL23747479 0.88 SMN1; SMN2 (0.58) MCHR1RAB9ANPC1POLBNAMPT
SCHEMBL23747483 0.88 SMN1; SMN2 (0.58) MCHR1RAB9ANPC1POLBNAMPT
SCHEMBL23747670 0.85 CHRM1 (0.57) CHRM1HTR2AMCHR1RAB9ANPC1
SCHEMBL23747395 0.85 CHRM1 (0.57) CHRM1HTR2AMCHR1RAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230133132-A1 NAMPT MODULATORS CYTOKINETICS, INC. 2023-05-04 US disclosed
US-20230133132-A1 NAMPT MODULATORS CYTOKINETICS, INC. 2023-05-04 US disclosed
US-20230133132-A1 NAMPT MODULATORS CYTOKINETICS, INC. 2023-05-04 US disclosed
CN-115515934-A NAMPT modulators 赛特凯恩蒂克公司 2022-12-23 CN disclosed
EP-4100393-A1 NAMPT MODULATORS Cytokinetics, Inc. (US) 2022-12-14 EP disclosed
WO-2021159015-A1 NAMPT MODULATORS CYTOKINETICS, INC. (US) 2021-08-12 WO disclosed
WO-2021159015-A1 NAMPT MODULATORS CYTOKINETICS, INC. (US) 2021-08-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230133132-A1 NAMPT MODULATORS NAMPT, MC4R, SIRT1 CHRM1 1155/4885HTR2A 2115/4885MCHR1 358/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.