SCHEMBL23732307

SCHEMBL23732307

O=C(O)c1cnn2ccc(N3CCOC[C@@H]3c3cc(F)cnc3O)nc12

nearest known ligand 0.54

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 19/20 0.54
ROS1 P08922 1/20 0.54
CYP2C9 P11712 1/20 0.54
CYP2C19 P33261 1/20 0.54
KCNH2 Q12809 1/20 0.54
NTRK3 Q16288 1/20 0.54
ALK Q9UM73 1/20 0.54
JAK2 O60674 15/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21911083 1.00 NTRK1 (0.54) NTRK1ROS1CYP2C9CYP2C19KCNH2
SCHEMBL21911084 0.92 NTRK1 (0.56) NTRK1JAK2
SCHEMBL24168768 0.88 NTRK1 (0.51) NTRK1ROS1CYP2C9CYP2C19KCNH2
SCHEMBL24030442 0.88 NTRK1 (0.65) NTRK1JAK2
SCHEMBL24030249 0.87 NTRK1 (0.64) NTRK1JAK2
SCHEMBL23149413 0.86 NTRK1 (0.70) NTRK1JAK2
SCHEMBL24168607 0.86 NTRK1 (0.68) NTRK1JAK2
SCHEMBL23732305 0.86 NTRK1 (0.67) NTRK1ROS1CYP2C9CYP2C19KCNH2
SCHEMBL23732308 0.86 NTRK1 (0.63) NTRK1JAK2
SCHEMBL21911499 0.83 NTRK1 (0.46) NTRK1JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3858834-A1 PYRAZOLOPYRIMIDINE DERIVATIVE AS SELECTIVE TRK INHIBITOR Shandong Luye Pharmaceutical Co., Ltd. (CN) 2021-08-04 EP disclosed