SCHEMBL23735162

SCHEMBL23735162

Cc1cc(I)c2c(c1F)CCNC2

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PNMT P11086 5/20 0.37
HTR6 P50406 5/20 0.34
ADRA2A P08913 1/20 0.33
ADRA2B P18089 1/20 0.33
ADRA2C P18825 1/20 0.33
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
PARP1 P09874 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19684784 0.84 PNMT (0.40) PNMTHTR6PARP1
SCHEMBL19711557 0.82 PNMT (0.39) PNMTHTR6ADRA2AADRA2BADRA2C
SCHEMBL19710968 0.80 PNMT (0.35) PNMTHTR6ADRA2AADRA2BADRA2C
SCHEMBL19711571 0.79 PNMT (0.49) PNMTHTR6ADRA2AADRA2BADRA2C
SCHEMBL19710976 0.79 PNMT (0.37) PNMTADRA2AADRA2BADRA2CHTR2A
SCHEMBL19710964 0.79 HTR2A (0.41) PNMTHTR6ADRA2AADRA2BADRA2C
SCHEMBL19710972 0.78 PNMT (0.33) PNMTHTR2AHTR2C
SCHEMBL23735224 0.77 HTR2C (0.35) PNMTHTR6ADRA2AADRA2BADRA2C
SCHEMBL20778128 0.77 PNMT (0.35) PNMTHTR6PARP1
SCHEMBL19678859 0.77 HTR2A (0.35) PNMTHTR6HTR2AHTR2CPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3464249-B1 SUBSTITUTED CARBONUCLEOSIDE DERIVATIVES USEFUL AS ANTICANCER AGENTS PFIZER (US) 2021-08-11 EP disclosed