SCHEMBL2373929

SCHEMBL2373929

CCCCc1csc(N)n1

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 2/20 0.53
SMN1; SMN2 Q16637 5/20 0.49
GABRA5 P31644 1/20 0.47
GABRB2 P47870 1/20 0.47
HSD17B10 Q99714 1/20 0.47
RAB9A P51151 4/20 0.46
NOS2 P35228 1/20 0.46
NPC1 O15118 3/20 0.44
ALDH1A1 P00352 2/20 0.44
ATM Q13315 1/20 0.44
AOC3 Q16853 1/20 0.43
MAPT P10636 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL44477 0.94 NOS1 (0.51) NOS1SMN1; SMN2GABRA5GABRB2HSD17B10
SCHEMBL9729165 0.92 NOS1 (0.50) NOS1SMN1; SMN2GABRA5GABRB2HSD17B10
SCHEMBL11588307 0.92 NOS1 (0.50) NOS1SMN1; SMN2GABRA5GABRB2HSD17B10
Ammonia Solution, Strong SCHEMBL28007740 0.92 NOS1 (0.50) NOS1SMN1; SMN2GABRA5GABRB2HSD17B10
SCHEMBL14643881 0.92 NOS1 (0.50) NOS1SMN1; SMN2GABRA5GABRB2HSD17B10
SCHEMBL3828155 0.92 NOS1 (0.50) NOS1SMN1; SMN2GABRA5GABRB2HSD17B10
Pyridine SCHEMBL27812107 0.88 NOS1 (0.51) NOS1SMN1; SMN2GABRA5GABRB2HSD17B10
SCHEMBL5911714 0.88
Pyridine SCHEMBL27812133 0.87 NOS1 (0.50) NOS1SMN1; SMN2GABRA5GABRB2HSD17B10
Toluene SCHEMBL27832196 0.87 NOS1 (0.58) NOS1SMN1; SMN2GABRA5GABRB2HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 77 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101648925-A 5-(4-chlorophenylmethyl)-4-tert-butyl-2-aminothiazolehydrobromate chiral crystal structure and preparation method thereof UNIV HUNAN 2010-02-17 CN claimed
CN-101492426-A Thiazole schiff base containing nitryl, preparation and uses thereof UNIV HUNAN (CN) 2009-07-29 CN claimed
CN-110279726-A Composition and its application containing Saxifragaceae Herba Chrysosplenii delavayi extract 嘉兴市爵拓科技有限公司 2019-09-27 CN disclosed
CN-104903320-B Nitrogen-containing heterocycle compound or its salt 富士胶片株式会社 2018-11-13 CN disclosed
CN-108685911-A 2-[(4- tertiary butyl thiazole -2- bases) Ya Anji ]Application of the thiazolin 4 one in pharmacy 山东大学 2018-10-23 CN disclosed
CN-106032365-B Benzal thiazolinone of 2 (base of thiazole 2) imino group 5 and preparation method and application 湖南大学 2018-03-23 CN disclosed
CN-105985298-B 2 [(base of 5 halogen thiazole 2) imino group] 5 benzal thiazolinones and preparation method and application 湖南大学 2018-02-23 CN disclosed
CN-105026386-B Antiviral compound 弗·哈夫曼-拉罗切有限公司 2017-08-01 CN disclosed
CN-106032365-A 2-(thiazol-2-yl)imino-5-(benzylidene)thiazolidin-4-one, and preparing method and applications thereof 湖南大学 2016-10-19 CN disclosed
CN-105026386-A Antiviral compounds HOFFMANN LA ROCHE 2015-11-04 CN disclosed
EP-1812433-B1 IMIDAZO[4,5-B]PYRIDIN-2-ONE AND OXAZOLO[4,5-B]PYRIDIN-2-ONE COMPOUNDS AND ANALOGS THEREOF AS THERAPEUTIC COMPOUNDS CANCER REC TECH LTD (GB) 2015-07-22 EP disclosed
CN-1069882-A The Compounds and methods for that suppresses HIV and correlated virus MEDIVIR AB (CH) 1993-03-17 CN disclosed
WO-1993003022-A1 COMPOUNDS AND METHODS FOR INHIBITION OF HIV AND RELATED VIRUSES MEDIVIR AB (SE) 1993-02-18 WO disclosed
US-4535081-A Antiallergic and antiulcer 1-oxo-1H-thiazolo[3,2-a]pyrimidine-2-carboxamides and intermediates therefor PFIZER INC. (US) 1985-08-13 US disclosed
US-4423048-A Antiallergic and antiulcer 1-oxo-1H-thiazolo[3,2-a]pyrimidine-2-carboxamides and intermediates therefor PFIZER INC. (US) 1983-12-27 US disclosed
US-4414388-A ANTIALLERGENS, ANTIULCER AGENTS PFIZER INC. (US) 1983-11-08 US disclosed
US-4321372-A Antiulcer thiazol-2-ylcarbamoyl-carboxylic acids, esters and amides PFIZER INC. (US) 1982-03-23 US disclosed
US-4277396-A FOR POLYACRYLONITRILE AND ACID-MODIFIED POLYAMIDES AND POLYESTERS BAYER AKTIENGESELLSCHAFT (DE) 1981-07-07 US disclosed
US-4104268-A POLYACRYLONITRILE, POLYESTERS, POLYAMIDES BAYER AKTIENGESELLSCHAFT (DE) 1978-08-01 US disclosed
US-4006127-A Cationic diazacyanine dyestuffs BAYER AKTIENGESELLSCHAFT (DT) 1977-02-01 US disclosed