SCHEMBL23748150

SCHEMBL23748150

C=CCCc1cc(F)c(F)cc1C(O)c1ccccn1

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.39
RECQL P46063 1/20 0.33
PRKDC P78527 1/20 0.33
KCNH2 Q12809 1/20 0.33
BRD4 O60885 1/20 0.32
KDM4E B2RXH2 1/20 0.31
TP53 P04637 1/20 0.30
SQOR Q9Y6N5 1/20 0.30
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23748219 0.86 F2RL1 (0.43) MAPTRECQLPRKDCKCNH2BRD4
SCHEMBL23748146 0.85 SQOR (0.30) SQORTSHR
SCHEMBL23748161 0.83 MAPT (0.43) MAPTRECQLKCNH2BRD4KDM4E
SCHEMBL23748230 0.79 MAPT (0.39) MAPTRECQLPRKDCKCNH2KDM4E
SCHEMBL23748295 0.74 F2RL1 (0.33) SQOR
SCHEMBL23748188 0.72 MAPT (0.41) MAPTKDM4ESQORTSHR
SCHEMBL23748168 0.72 MAPT (0.44) MAPTRECQLKCNH2KDM4ETSHR
SCHEMBL23748213 0.69 LIG1 (0.43) MAPTKDM4ETSHR
SCHEMBL23748227 0.69 SLC6A2 (0.33) MAPTKCNH2TSHR
SCHEMBL23748201 0.69 CTSA (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230002409-A1 MACROCYCLIC FLU ENDONUCLEASE INHIBITORS JANSSEN BIOPHARMA INC (US) 2023-01-05 US disclosed
US-11312727-B1 Macrocyclic flu endonuclease inhibitors Janssen Biopharma, Inc. (US) 2022-04-26 US disclosed
EP-3864020-A1 MACROCYCLIC FLU ENDONUCLEASE INHIBITORS Janssen BioPharma, Inc. (US) 2021-08-18 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230002409-A1 MACROCYCLIC FLU ENDONUCLEASE INHIBITORS ACE, PNP, FEN1 MAPT 2999/4885RECQL 243/4885PRKDC 477/4885
US-11312727-B1 Macrocyclic flu endonuclease inhibitors ACE, FEN1, PNP MAPT 3026/4885RECQL 134/4885PRKDC 667/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.