SCHEMBL23768898

SCHEMBL23768898

OCc1cn(Cc2ccc(N3CC4(CC4)C3)nc2)cn1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 3/20 0.49
KDM4E B2RXH2 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
ALDH1A1 P00352 3/20 0.34
HPGD P15428 3/20 0.34
HSD17B10 Q99714 3/20 0.34
TSHR P16473 2/20 0.34
HIF1A Q16665 2/20 0.34
CYP2D6 P10635 1/20 0.34
BTK Q06187 2/20 0.33
PHF8 Q9UPP1 1/20 0.32
CYP1A2 P05177 1/20 0.32
SMO Q99835 1/20 0.31
CPB2 Q96IY4 1/20 0.31
USP2 O75604 1/20 0.30
RET P07949 1/20 0.30
TNIK Q9UKE5 1/20 0.30
KCNJ1 P48048 3/20 0.30
CACNA1G O43497 1/20 0.30
CACNA1H O95180 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21736669 0.81 KLKB1 (0.56) KLKB1ALDH1A1HPGDHSD17B10TSHR
SCHEMBL21713011 0.80 SMO (0.43) KLKB1ALDH1A1HPGDHSD17B10TSHR
SCHEMBL29906615 0.80 SMO (0.43) KLKB1ALDH1A1HPGDHSD17B10TSHR
SCHEMBL22166237 0.78 KLKB1 (0.56) KLKB1ALDH1A1HPGDHSD17B10TSHR
SCHEMBL21736897 0.76 KLKB1 (0.56) KLKB1KDM4EALDH1A1HPGDHSD17B10
Trifluoroacetic Acid SCHEMBL23830228 0.76 KLKB1 (0.52) KLKB1ALDH1A1HPGDHSD17B10TSHR
Trifluoroacetic Acid SCHEMBL29906622 0.76 KLKB1 (0.52) KLKB1ALDH1A1HPGDHSD17B10TSHR
SCHEMBL23830229 0.74 KLKB1 (0.52) KLKB1ALDH1A1HPGDHSD17B10TSHR
SCHEMBL23769680 0.74 KLKB1 (0.40) KLKB1KDM4EL3MBTL1ALDH1A1HPGD
SCHEMBL23769373 0.69 BTK (0.51) KLKB1L3MBTL1HSD17B10BTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021160718-A1 HETEROAROMATIC CARBOXAMIDE DERIVATIVES AS PLASMA KALLIKREIN INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2021-08-19 WO disclosed