SCHEMBL23768926

SCHEMBL23768926

CCOC(=O)c1cc(C(O)c2ccc(N3CC(C)C(F)(F)C3)nc2CC)nn1C(C)C

nearest known ligand 0.31

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CCR4 P51679 1/20 0.31
KDM4E B2RXH2 1/20 0.30
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30
RXFP1 Q9HBX9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30087456 0.88 CCR4 (0.31) CCR4
SCHEMBL23754333 0.88 CCR4 (0.31) CCR4
SCHEMBL23769535 0.83 NPC1 (0.30) KDM4ENPC1RAB9ARXFP1
SCHEMBL23769707 0.78 FAAH (0.34) KDM4ENPC1RAB9ARXFP1
SCHEMBL29906659 0.75 KLKB1 (0.31) KDM4ENPC1RAB9ARXFP1
SCHEMBL29906628 0.75 KLKB1 (0.31) KDM4ENPC1RAB9ARXFP1
SCHEMBL23769712 0.75 KLKB1 (0.34) CCR4KDM4ENPC1RAB9ARXFP1
SCHEMBL23769467 0.72 ITGAL (0.31)
SCHEMBL23769529 0.70 KLKB1 (0.33)
SCHEMBL23843236 0.69 KLKB1 (0.45) RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021160718-A1 HETEROAROMATIC CARBOXAMIDE DERIVATIVES AS PLASMA KALLIKREIN INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2021-08-19 WO disclosed