SCHEMBL23769225

SCHEMBL23769225

CC(C)(C)c1nc(N2CC3CC3C2)ccc1Cn1cc(C(=O)O)cn1

nearest known ligand 0.52

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BTK Q06187 11/20 0.52
KLKB1 P03952 8/20 0.48
L3MBTL1 Q9Y468 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23769337 0.93 BTK (0.51) BTKKLKB1L3MBTL1
SCHEMBL18818263 0.90 BTK (0.62) BTKKLKB1L3MBTL1
SCHEMBL23843098 0.89 BTK (0.49) BTKKLKB1L3MBTL1
SCHEMBL30140684 0.86 KLKB1 (0.61) BTKKLKB1
SCHEMBL20541004 0.86 KLKB1 (0.61) BTKKLKB1
SCHEMBL23769242 0.85 BTK (0.49) BTKKLKB1
SCHEMBL23769217 0.84 KLKB1 (0.49) BTKKLKB1L3MBTL1
SCHEMBL23768875 0.84 KLKB1 (0.48) BTKKLKB1
SCHEMBL23768857 0.84 KLKB1 (0.48) BTKKLKB1L3MBTL1
SCHEMBL23769334 0.83 KLKB1 (0.47) BTKKLKB1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021160718-A1 HETEROAROMATIC CARBOXAMIDE DERIVATIVES AS PLASMA KALLIKREIN INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2021-08-19 WO disclosed