SCHEMBL23769302

SCHEMBL23769302

CCOC(=O)c1cc(Cc2ccc(N3CC4[C@H](C3)C4(F)F)nc2/C=C/c2ccccc2)no1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 5/20 0.34
ALDH1A1 P00352 3/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
L3MBTL1 Q9Y468 2/20 0.34
KDM4E B2RXH2 1/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
XBP1 P17861 1/20 0.34
TRPA1 O75762 1/20 0.32
PDE10A Q9Y233 1/20 0.32
DHFR P00374 1/20 0.32
TMIGD3 P0DMS9 1/20 0.32
LMNA P02545 1/20 0.32
ALOX12 P18054 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2C19 P33261 1/20 0.32
HSD17B10 Q99714 1/20 0.32
ADORA2B P29275 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23843116 1.00 ADORA3 (0.34) ADORA3ALDH1A1MEN1KMT2AL3MBTL1
SCHEMBL23769304 0.89 KLKB1 (0.39) ADORA3ALDH1A1MEN1KMT2AL3MBTL1
SCHEMBL23768962 0.88 KLKB1 (0.34) MAPTTRPA1PDE10ALMNAADORA2B
SCHEMBL23769694 0.85 KLKB1 (0.39) ALDH1A1KMT2AKDM4EHPGDTRPA1
SCHEMBL23769464 0.84 KLKB1 (0.33) ALDH1A1MEN1KMT2AL3MBTL1TRPA1
SCHEMBL23769506 0.84 MAPT (0.34) ALDH1A1KDM4EMAPTHPGDTRPA1
SCHEMBL23769297 0.83 KLKB1 (0.34) ALDH1A1MEN1KMT2AL3MBTL1KDM4E
SCHEMBL23769405 0.82 KLKB1 (0.40) KDM4ETRPA1PDE10AHSD17B10
SCHEMBL23843172 0.78 PDE10A (0.33) ALDH1A1MEN1KMT2AL3MBTL1PDE10A
SCHEMBL23768964 0.77 KLKB1 (0.41) KDM4EMAPTTRPA1PDE10ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021160718-A1 HETEROAROMATIC CARBOXAMIDE DERIVATIVES AS PLASMA KALLIKREIN INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2021-08-19 WO disclosed