SCHEMBL23769308

SCHEMBL23769308

CCOC(=O)c1cn(Cc2ccc(N3CC4[C@H](C3)C4(F)F)nc2CO)nn1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
LMNA P02545 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.43
HPGD P15428 1/20 0.43
KLKB1 P03952 7/20 0.40
GLA P06280 1/20 0.39
MAPK1 P28482 2/20 0.38
MEN1 O00255 1/20 0.36
TSHR P16473 1/20 0.36
KMT2A Q03164 1/20 0.36
TP53 P04637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23754180 1.00 ALDH1A1 (0.46) ALDH1A1LMNASMN1; SMN2HPGDKLKB1
SCHEMBL31357759 1.00 ALDH1A1 (0.46) ALDH1A1LMNASMN1; SMN2HPGDKLKB1
SCHEMBL23769285 0.94 ALDH1A1 (0.47) ALDH1A1LMNASMN1; SMN2HPGDKLKB1
SCHEMBL23469650 0.90 ALDH1A1 (0.48) ALDH1A1LMNASMN1; SMN2HPGDKLKB1
SCHEMBL30140712 0.90 ALDH1A1 (0.48) ALDH1A1LMNASMN1; SMN2HPGDKLKB1
SCHEMBL23769183 0.90 ALDH1A1 (0.48) ALDH1A1LMNASMN1; SMN2HPGDKLKB1
SCHEMBL23769177 0.88 ALDH1A1 (0.49) ALDH1A1LMNASMN1; SMN2HPGDKLKB1
SCHEMBL23769141 0.88 ALDH1A1 (0.49) ALDH1A1LMNASMN1; SMN2HPGDKLKB1
SCHEMBL23754188 0.88 ALDH1A1 (0.48) ALDH1A1LMNASMN1; SMN2HPGDKLKB1
SCHEMBL23768900 0.88 ALDH1A1 (0.48) ALDH1A1LMNASMN1; SMN2HPGDKLKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021160718-A1 HETEROAROMATIC CARBOXAMIDE DERIVATIVES AS PLASMA KALLIKREIN INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2021-08-19 WO disclosed