SCHEMBL23769317

SCHEMBL23769317

CCOC(=O)c1cn(Cc2cnc(N3CC4C[C@H]4C3)cc2C(F)(F)F)cn1

nearest known ligand 0.44

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BTK Q06187 8/20 0.44
KLKB1 P03952 6/20 0.41
RBP4 P02753 3/20 0.35
NOTUM Q6P988 1/20 0.34
HPGD P15428 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23773116 1.00 BTK (0.44) BTKKLKB1RBP4NOTUMHPGD
SCHEMBL23769202 0.88 BTK (0.42) BTKKLKB1NOTUM
SCHEMBL23768861 0.87 BTK (0.47) BTKKLKB1RBP4
SCHEMBL23769320 0.86 NOTUM (0.42) BTKKLKB1NOTUMKMT2A
SCHEMBL18795065 0.85 BTK (0.57) BTKKLKB1HPGDSMN1; SMN2
SCHEMBL18815275 0.82 BTK (0.57) BTKKLKB1
SCHEMBL21736670 0.80 KLKB1 (0.56) BTKKLKB1NOTUMHPGDSMN1; SMN2
SCHEMBL23769406 0.79 KLKB1 (0.48) KLKB1NOTUMKMT2A
SCHEMBL23769313 0.79 KLKB1 (0.48) KLKB1NOTUMHPGDKMT2A
SCHEMBL23769142 0.79 KLKB1 (0.44) KLKB1RBP4NOTUMKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021160718-A1 HETEROAROMATIC CARBOXAMIDE DERIVATIVES AS PLASMA KALLIKREIN INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2021-08-19 WO disclosed