SCHEMBL23769377

SCHEMBL23769377

CCc1nc(N2CC3CC3C2)ccc1CCCOC

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 5/20 0.34
SMPD3 Q9NY59 2/20 0.33
HCRTR1 O43613 1/20 0.31
HCRTR2 O43614 1/20 0.31
RET P07949 1/20 0.31
PDE10A Q9Y233 1/20 0.31
HSD11B1 P28845 1/20 0.30
REN P00797 3/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23769583 0.96 SMPD3 (0.34) KLKB1SMPD3HCRTR1HCRTR2RET
SCHEMBL23843150 0.92 KLKB1 (0.35) KLKB1SMPD3HCRTR1HCRTR2RET
SCHEMBL23768950 0.82 SMPD3 (0.39) KLKB1SMPD3HCRTR1HCRTR2PDE10A
SCHEMBL23769616 0.79 SMPD3 (0.36) KLKB1SMPD3HCRTR1HCRTR2PDE10A
SCHEMBL23843137 0.79 KLKB1 (0.35) KLKB1SMPD3HCRTR1HCRTR2PDE10A
SCHEMBL23769134 0.77 KLKB1 (0.38) KLKB1HCRTR1HCRTR2
SCHEMBL23754018 0.75 SMPD3 (0.34) KLKB1SMPD3HCRTR1HCRTR2PDE10A
SCHEMBL29906555 0.75 SMPD3 (0.34) KLKB1SMPD3HCRTR1HCRTR2PDE10A
SCHEMBL23769391 0.75 SMPD3 (0.34) KLKB1SMPD3HCRTR1HCRTR2RET
SCHEMBL23830202 0.74 KLKB1 (0.39) KLKB1SMPD3HCRTR1HCRTR2HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021160718-A1 HETEROAROMATIC CARBOXAMIDE DERIVATIVES AS PLASMA KALLIKREIN INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2021-08-19 WO disclosed