SCHEMBL23769691

SCHEMBL23769691

CC(=O)N/N=C/c1ccc(N2CC(C)C(F)(F)C2)nc1C

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GFER P55789 2/20 0.34
KDM4E B2RXH2 5/20 0.33
ALDH1A1 P00352 4/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
LMNA P02545 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
USP2 O75604 1/20 0.32
ACACB O00763 1/20 0.32
HPGD P15428 3/20 0.31
BACE1 P56817 2/20 0.31
BCHE P06276 1/20 0.31
ACHE P22303 1/20 0.31
NPC1 O15118 2/20 0.30
GBA1 P04062 2/20 0.30
GAA P10253 2/20 0.30
HTT P42858 1/20 0.30
RAB9A P51151 1/20 0.30
MAPT P10636 1/20 0.30
P2RX7 Q99572 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23753983 0.84 KLKB1 (0.37) GFERKDM4EALDH1A1MEN1KMT2A
SCHEMBL29906540 0.84 KLKB1 (0.37) GFERKDM4EALDH1A1MEN1KMT2A
SCHEMBL23753981 0.84 KLKB1 (0.37) GFERKDM4EALDH1A1MEN1KMT2A
SCHEMBL23768952 0.80 GFER (0.38) GFERKDM4EALDH1A1MEN1KMT2A
SCHEMBL23769214 0.70 MAP3K12 (0.30)
SCHEMBL8802519 0.68 KDM4E (0.44) KDM4EALDH1A1MEN1KMT2ALMNA
SCHEMBL8802527 0.68 KDM4E (0.44) KDM4EALDH1A1MEN1KMT2ALMNA
SCHEMBL23768790 0.66 KLKB1 (0.36)
SCHEMBL24918819 0.66 KLKB1 (0.48)
SCHEMBL21861490 0.63 ACACB (0.37) ACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021160718-A1 HETEROAROMATIC CARBOXAMIDE DERIVATIVES AS PLASMA KALLIKREIN INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2021-08-19 WO disclosed