SCHEMBL29906540

SCHEMBL29906540

CC(=O)N/N=C/c1ccc(N2CC3C(C2)C3(F)F)nc1C

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 9/20 0.37
GFER P55789 2/20 0.36
KDM4E B2RXH2 3/20 0.34
ALDH1A1 P00352 2/20 0.34
LMNA P02545 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
MEN1 O00255 1/20 0.34
USP2 O75604 1/20 0.34
KMT2A Q03164 1/20 0.34
ACACB O00763 2/20 0.33
HPGD P15428 1/20 0.32
NPC1 O15118 1/20 0.32
GBA1 P04062 1/20 0.32
HTT P42858 1/20 0.32
GRM4 Q14833 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23753983 1.00 KLKB1 (0.37) KLKB1GFERKDM4EALDH1A1LMNA
SCHEMBL23753981 1.00 KLKB1 (0.37) KLKB1GFERKDM4EALDH1A1LMNA
SCHEMBL23768952 0.85 GFER (0.38) KLKB1GFERKDM4EALDH1A1LMNA
SCHEMBL23769691 0.84 GFER (0.34) GFERKDM4EALDH1A1LMNASMN1; SMN2
SCHEMBL31033243 0.78 KLKB1 (0.36) KLKB1GFERKDM4EALDH1A1MEN1
SCHEMBL21713091 0.78 KLKB1 (0.36) KLKB1GFERKDM4EALDH1A1MEN1
SCHEMBL29906594 0.73 KLKB1 (0.46) KLKB1ACACB
SCHEMBL23754000 0.73 KLKB1 (0.46) KLKB1ACACB
SCHEMBL23843164 0.72 KLKB1 (0.37) KLKB1KDM4EALDH1A1
SCHEMBL8802519 0.70 KDM4E (0.44) KDM4EALDH1A1LMNAMEN1USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116120287-B Heteroaromatic carboxamide derivatives as inhibitors of plasma kallikrein 勃林格殷格翰国际有限公司 2025-01-28 CN disclosed
CN-116120287-A Heteroaromatic carboxamide derivatives as inhibitors of plasma kallikrein 勃林格殷格翰国际有限公司 2023-05-16 CN disclosed
CN-115052873-A Heteroaromatic carboxamide derivatives as plasma kallikrein inhibitors 勃林格殷格翰国际有限公司 2022-09-13 CN disclosed