SCHEMBL23770979

SCHEMBL23770979

CC(C)(C)OC(=O)Nc1cncc(Nc2cccnn2)c1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 2/20 0.50
CYP17A1 P05093 4/20 0.41
SYK P43405 1/20 0.39
RAB9A P51151 1/20 0.39
BRD4 O60885 2/20 0.38
BCL2 P10415 1/20 0.38
JAK2 O60674 3/20 0.38
JAK1 P23458 3/20 0.38
TYK2 P29597 2/20 0.38
TOP2A P11388 1/20 0.37
TOP2B Q02880 1/20 0.37
LCK P06239 1/20 0.36
JAK3 P52333 1/20 0.36
ATR Q13535 1/20 0.36
AURKA O14965 1/20 0.36
AURKB Q96GD4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30196114 1.00 NAMPT (0.50) NAMPTCYP17A1SYKRAB9ABRD4
SCHEMBL23771038 0.84 NAMPT (0.48) NAMPTCYP17A1SYKRAB9ATOP2A
SCHEMBL22574157 0.81 JAK2 (0.43) NAMPTRAB9AJAK2JAK1TYK2
SCHEMBL31038470 0.80 NAMPT (0.46) NAMPTCYP17A1RAB9AJAK2JAK1
SCHEMBL4093611 0.80 NAMPT (0.46) NAMPTCYP17A1RAB9AJAK2JAK1
SCHEMBL14428036 0.80 NAMPT (0.54) NAMPTCYP17A1SYKRAB9ATOP2A
SCHEMBL6756707 0.75 NAMPT (0.60) NAMPTCYP17A1RAB9ABCL2
SCHEMBL29674394 0.75 NAMPT (0.49) NAMPTCYP17A1SYKTOP2ATOP2B
SCHEMBL349933 0.75 NAMPT (0.80) NAMPTRAB9A
SCHEMBL12735928 0.75 NAMPT (0.49) NAMPTCYP17A1SYKTOP2ATOP2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3728217-B1 CHROMENOPYRIDINE DERIVATIVES AS PHOSPHATIDYLINOSITOL PHOSPHATE KINASE INHIBITORS HIBERCELL INC (US) 2023-11-15 EP disclosed
US-11584763-B2 Chromenopyridine derivatives as phosphatidylinositol phosphate kinase inhibitors HIBERCELL, INC. (US) 2023-02-21 US disclosed
US-11535635-B2 2022-12-27 US disclosed
US-20210253600-A1 CHROMENOPYRIDINE DERIVATIVES AS PHOSPHATIDYLINOSITOL PHOSPHATE KINASE INHIBITORS HIBERCELL, INC. 2021-08-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11584763-B2 Chromenopyridine derivatives as phosphatidylinositol phosphate kinase inhibitors PIP5K1A, PIP5K1B, PI4KA NAMPT 1015/4885CYP17A1 3667/4885SYK 2210/4885
US-11535635-B2 PIP5K1A, PI4K2A, PIP5K1B NAMPT 766/4885CYP17A1 1438/4885SYK 4559/4885
US-20210253600-A1 CHROMENOPYRIDINE DERIVATIVES AS PHOSPHATIDYLINOSITOL PHOSPHATE KINASE INHIBITORS PIP5K1A, PIP5K1B, PI4KA NAMPT 1015/4885CYP17A1 3667/4885SYK 2210/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.