SCHEMBL23778232

SCHEMBL23778232

COc1ccc(C2(C#N)CCC(N3CCCN(C(=O)O)CC3)CC2)nc1

nearest known ligand 0.44

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 16/20 0.44
KCNH2 Q12809 1/20 0.41
PKM P14618 1/20 0.39
IRAK4 Q9NWZ3 1/20 0.39
ALDH1A1 P00352 1/20 0.38
TSHR P16473 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23778420 0.91 HRH3 (0.40) HRH3KCNH2ALDH1A1
SCHEMBL20066025 0.89 HRH3 (0.46) HRH3PKMIRAK4ALDH1A1
SCHEMBL20066227 0.88 HRH3 (0.45) HRH3KCNH2IRAK4ALDH1A1
SCHEMBL23778350 0.87 HRH3 (0.39) HRH3KCNH2IRAK4
SCHEMBL20066036 0.86 HRH3 (0.43) HRH3KCNH2IRAK4ALDH1A1
SCHEMBL20066037 0.85 HRH3 (0.43) HRH3KCNH2IRAK4ALDH1A1TSHR
SCHEMBL23778387 0.85 HRH3 (0.43) HRH3KCNH2
SCHEMBL23778451 0.85 HRH3 (0.40) HRH3KCNH2IRAK4
SCHEMBL23778281 0.85 HRH3 (0.45) HRH3KCNH2
SCHEMBL23778270 0.85 ALDH1A1 (0.46) HRH3PKMALDH1A1TSHRKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3526207-B1 HETEROCYCLIC COMPOUNDS HAVING ACTIVITY AS MODULATORS OF MUSCARINIC M1 AND/OR M4 RECEPTORS IN THE TREATMENT OF CNS DISEASES AND PAINS. HEPTARES THERAPEUTICS LTD (GB) 2021-09-08 EP claimed