SCHEMBL23795705

SCHEMBL23795705

Cc1ccc(C(=O)O)cc1-c1ccc2nc(NC(=O)C3CC3)cn2c1

nearest known ligand 0.63

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 19/20 0.63
ABL1 P00519 4/20 0.58
MAPK13 O15264 1/20 0.56
BRAF P15056 1/20 0.56
KDR P35968 1/20 0.56
MAPK12 P53778 1/20 0.56
MAPK11 Q15759 1/20 0.56
MAPK14 Q16539 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23795720 0.90 LRRK2 (0.61) LRRK2ABL1MAPK13BRAFKDR
SCHEMBL25540594 0.89 LRRK2 (0.77) LRRK2ABL1
SCHEMBL22380363 0.86 LRRK2 (0.78) LRRK2ABL1
SCHEMBL22380088 0.85 LRRK2 (0.79) LRRK2ABL1MAPK13BRAFKDR
SCHEMBL22380094 0.84 LRRK2 (0.79) LRRK2ABL1MAPK13BRAFKDR
SCHEMBL23795682 0.83 LRRK2 (0.60) LRRK2ABL1
SCHEMBL25540591 0.82 LRRK2 (0.59) LRRK2ABL1KDR
SCHEMBL23795715 0.81 CSNK1D (0.56) ABL1KDR
SCHEMBL24012496 0.80 LRRK2 (0.81) LRRK2ABL1
SCHEMBL22362800 0.79 LRRK2 (0.79) LRRK2ABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230151001-A9 IMIDAZOPYRIDINE DERIVATIVES AND AZA-IMIDAZOPYRIDINE DERIVATIVES AS JANUS KINASE 2 INHIBITORS AND USES THEREOF DANA-FARBER CANCER INSTITUTE, INC. (US) 2023-05-18 US disclosed
US-20220127260-A1 IMIDAZOPYRIDINE DERIVATIVES AND AZA-IMIDAZOPYRIDINE DERIVATIVES AS JANUS KINASE 2 INHIBITORS AND USES THEREOF DANA-FARBER CANCER INSTITUTE, INC. (US) 2022-04-28 US disclosed
EP-3877371-A1 IMIDAZOPYRIDINE DERIVATIVES AND AZA-IMIDAZOPYRIDINE DERIVATIVES AS JANUS KINASE 2 INHIBITORS AND USES THEREOF Dana-Farber Cancer Institute, Inc. (US) 2021-09-15 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220127260-A1 IMIDAZOPYRIDINE DERIVATIVES AND AZA-IMIDAZOPYRIDINE DERIVATIVES AS JANUS KINASE 2 INHIBITORS AND USES THEREOF JAK1, JAK2, JAK3 LRRK2 2176/4885ABL1 16/4885MAPK13 162/4885
US-20230151001-A9 IMIDAZOPYRIDINE DERIVATIVES AND AZA-IMIDAZOPYRIDINE DERIVATIVES AS JANUS KINASE 2 INHIBITORS AND USES THEREOF JAK1, JAK2, JAK3 LRRK2 2176/4885ABL1 16/4885MAPK13 162/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.