SCHEMBL23798604

SCHEMBL23798604

CNC1CCN(C2CCC3(CC2)C(=O)Nc2ccccc23)C1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 3/20 0.47
OPRK1 P41145 3/20 0.47
OPRL1 P41146 3/20 0.47
BACE1 P56817 3/20 0.41
HTR1A P08908 9/20 0.40
HTR2A P28223 9/20 0.40
HTR7 P34969 9/20 0.40
HTR6 P50406 9/20 0.40
MAPK14 Q16539 1/20 0.39
TNKS O95271 1/20 0.37
TNKS2 Q9H2K2 1/20 0.37
CALCRL Q16602 1/20 0.37
PDK2 Q15119 1/20 0.35
PDK4 Q16654 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23798012 0.86 MAPK14 (0.45) MAPK14
SCHEMBL23778419 0.85 BACE1 (0.44) OPRM1OPRK1OPRL1BACE1HTR1A
SCHEMBL23798606 0.84 OPRM1 (0.40) OPRM1OPRK1OPRL1HTR1AHTR2A
SCHEMBL23799157 0.84 HRH4 (0.37) OPRM1OPRK1OPRL1HTR7MAPK14
SCHEMBL23798696 0.83 HRH4 (0.36) OPRM1OPRK1OPRL1HTR1AHTR2A
SCHEMBL29709346 0.82 CHRM1 (0.45) OPRM1OPRK1OPRL1BACE1HTR1A
SCHEMBL20073883 0.82 CHRM1 (0.45) OPRM1OPRK1OPRL1BACE1HTR1A
SCHEMBL29709353 0.82 CHRM1 (0.45) OPRM1OPRK1OPRL1BACE1HTR1A
SCHEMBL20073879 0.82 CHRM1 (0.45) OPRM1OPRK1OPRL1BACE1HTR1A
SCHEMBL23798681 0.81 OPRM1 (0.47) OPRM1OPRK1OPRL1BACE1HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3526207-B1 HETEROCYCLIC COMPOUNDS HAVING ACTIVITY AS MODULATORS OF MUSCARINIC M1 AND/OR M4 RECEPTORS IN THE TREATMENT OF CNS DISEASES AND PAINS. HEPTARES THERAPEUTICS LTD (GB) 2021-09-08 EP disclosed