SCHEMBL23799161

SCHEMBL23799161

CN1CCC2(C1)CN(C1CCC(C#N)(c3ccccc3)CC1)C2

nearest known ligand 0.59

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.47
KDM1A O60341 1/20 0.45
OPRM1 P35372 6/20 0.44
DRD4 P21917 1/20 0.42
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30179321 0.82 CYP2D6 (0.49) CYP2D6KDM1AOPRM1
SCHEMBL23778300 0.82 CYP2D6 (0.50) CYP2D6KDM1AOPRM1KMT2A
SCHEMBL23798654 0.81 OPRL1 (0.56) CYP2D6KDM1AOPRM1KMT2A
SCHEMBL9435664 0.80 OPRL1 (0.58) CYP2D6KDM1AOPRM1
SCHEMBL20066074 0.78 CYP2D6 (0.47) CYP2D6KDM1AOPRM1KMT2A
SCHEMBL504355 0.76 OPRM1 (0.70) OPRM1KMT2A
SCHEMBL23778282 0.76 CYP2D6 (0.53) CYP2D6KDM1AOPRM1KMT2A
SCHEMBL13654981 0.76 OPRM1 (0.54) CYP2D6KDM1AOPRM1
SCHEMBL9435475 0.75 CYP2D6 (0.49) CYP2D6KDM1AOPRM1KMT2A
SCHEMBL6963361 0.75 CYP2D6 (0.49) CYP2D6KDM1AOPRM1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3526207-B1 HETEROCYCLIC COMPOUNDS HAVING ACTIVITY AS MODULATORS OF MUSCARINIC M1 AND/OR M4 RECEPTORS IN THE TREATMENT OF CNS DISEASES AND PAINS. HEPTARES THERAPEUTICS LTD (GB) 2021-09-08 EP disclosed