SCHEMBL23865256

SCHEMBL23865256

O=C1NCCc2ccc(-n3cnc(C4CC4)c3)cc21

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MAP3K5 Q99683 12/20 0.46
PARP1 P09874 6/20 0.46
PARP10 Q53GL7 6/20 0.46
F7 P08709 1/20 0.46
F3 P13726 1/20 0.46
MAPKAPK2 P49137 1/20 0.41
PDPK1 O15530 1/20 0.40
PARP11 Q9NR21 1/20 0.40
DDB1 Q16531 1/20 0.39
CRBN Q96SW2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20774424 0.89 MAP3K5 (0.46) MAP3K5DDB1CRBN
SCHEMBL28607413 0.81 MAP3K5 (0.38) MAP3K5PARP1PARP10F7F3
SCHEMBL22473965 0.81 PARP10 (0.41) MAP3K5PARP1PARP10F7F3
SCHEMBL21750535 0.80 MAP3K5 (0.38) MAP3K5DDB1CRBN
SCHEMBL20489212 0.80 MAP3K5 (0.49) MAP3K5PARP1PARP10PARP11
SCHEMBL29978642 0.80 MAP3K5 (0.49) MAP3K5PARP1PARP10PARP11
SCHEMBL28941273 0.80 PARP10 (0.40) MAP3K5PARP1PARP10F7F3
SCHEMBL28887761 0.80 PARP10 (0.40) MAP3K5PARP1PARP10F7F3
SCHEMBL30362996 0.80 PARP10 (0.40) MAP3K5PARP1PARP10F7F3
SCHEMBL30362908 0.79 GRM5 (0.38) MAP3K5PARP10PARP11DDB1CRBN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110294742-B Fused ring ASK1 inhibitor and application thereof 山东轩竹医药科技有限公司 2023-01-31 CN disclosed
EP-3572401-B1 ASK1 INHIBITOR AND PREPARATION METHOD AND USE THEREOF FUJIAN COSUNTER PHARMACEUTICAL CO LTD (CN) 2021-09-29 EP disclosed