SCHEMBL29978642

SCHEMBL29978642

Cc1cc2c(cc1-n1cnc(C3CC3)c1)C(=O)NCC2

nearest known ligand 0.49

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MAP3K5 Q99683 17/20 0.49
PARP10 Q53GL7 2/20 0.40
PARP11 Q9NR21 1/20 0.40
PARP1 P09874 1/20 0.40
KDM4E B2RXH2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20489212 1.00 MAP3K5 (0.49) MAP3K5PARP10PARP11PARP1KDM4E
SCHEMBL21705962 0.89 MAP3K5 (0.47) MAP3K5
SCHEMBL28607413 0.87 MAP3K5 (0.38) MAP3K5PARP10PARP11PARP1KDM4E
SCHEMBL22473965 0.87 PARP10 (0.41) MAP3K5PARP10PARP11PARP1KDM4E
SCHEMBL30362996 0.86 PARP10 (0.40) MAP3K5PARP10PARP11PARP1KDM4E
SCHEMBL28941273 0.86 PARP10 (0.40) MAP3K5PARP10PARP11PARP1KDM4E
SCHEMBL28887761 0.86 PARP10 (0.40) MAP3K5PARP10PARP11PARP1KDM4E
SCHEMBL28910942 0.84 MAP3K5 (0.39) MAP3K5PARP10PARP11PARP1KDM4E
SCHEMBL28533456 0.80 MAP3K5 (0.36) MAP3K5PARP10PARP11PARP1KDM4E
SCHEMBL28539135 0.80 MAP3K5 (0.38) MAP3K5PARP10PARP11PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115504986-B Apoptosis signal regulating kinase inhibitor and preparation method and application thereof 江苏豪森药业集团有限公司 2024-05-14 CN disclosed
CN-115504986-A Apoptosis signal regulating kinase inhibitor and preparation method and application thereof 江苏豪森药业集团有限公司 2022-12-23 CN disclosed
CN-111094250-B Apoptosis signal regulating kinase inhibitor and preparation method and application thereof 江苏豪森药业集团有限公司 2022-11-04 CN disclosed