SCHEMBL2390948

SCHEMBL2390948

CCOC(=O)/C=C/c1cc(Cl)cc(-c2ccc(OCc3ccccc3)c(C34CC5CC(CC(C5)C3)C4)c2)c1OCC

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC11 Q96DB2 4/20 0.40
PTPN11 Q06124 4/20 0.37
NR0B2 Q15466 2/20 0.37
PTGER1 P34995 4/20 0.37
PTGER4 P35408 1/20 0.37
PTGER3 P43115 1/20 0.37
PTGER2 P43116 1/20 0.37
S1PR1 P21453 1/20 0.37
HDAC2 Q92769 1/20 0.37
KDM4E B2RXH2 2/20 0.36
LMNA P02545 2/20 0.36
ALDH1A1 P00352 1/20 0.36
KCNA3 P22001 1/20 0.36
HDAC8 Q9BY41 2/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
CCNC P24863 1/20 0.35
CDK8 P49336 1/20 0.35
CYP2C9 P11712 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2390735 0.95 HDAC11 (0.40) HDAC11PTPN11NR0B2PTGER1PTGER4
SCHEMBL6022621 0.93 HDAC11 (0.47) HDAC11PTPN11NR0B2PTGER1PTGER4
SCHEMBL6022615 0.93 HDAC11 (0.47) HDAC11PTPN11NR0B2PTGER1PTGER4
SCHEMBL6022897 0.86 HDAC11 (0.47) HDAC11PTPN11NR0B2PTGER1PTGER4
SCHEMBL6022901 0.86 HDAC11 (0.47) HDAC11PTPN11NR0B2PTGER1PTGER4
SCHEMBL2391779 0.86 HDAC11 (0.45) HDAC11PTPN11NR0B2S1PR1HDAC2
SCHEMBL2390957 0.86 HDAC11 (0.45) HDAC11PTPN11NR0B2S1PR1HDAC2
SCHEMBL2391835 0.86 PTPN11 (0.48) HDAC11PTPN11NR0B2HDAC2KDM4E
SCHEMBL2390953 0.85 PSEN1 (0.37) HDAC11PTPN11NR0B2PTGER1S1PR1
SCHEMBL2392575 0.84 PTPN11 (0.55) HDAC11PTPN11NR0B2HDAC2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE42700-E1 Induction of apoptosis in cancer cells SANFORD-BURNHAM MEDICAL RESEARCH INSTITUTE (US) 2011-09-13 US disclosed