SCHEMBL23917286

SCHEMBL23917286

C=CC(=O)c1cc(F)cc(-c2n[nH]c3ncnc(N)c23)c1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 6/20 0.41
FGFR4 P22455 5/20 0.41
MAP4K4 O95819 9/20 0.40
FGFR2 P21802 5/20 0.38
FGFR3 P22607 5/20 0.38
EGFR P00533 3/20 0.35
PIK3CD O00329 2/20 0.35
ABL1 P00519 2/20 0.35
HCK P08631 2/20 0.35
SRC P12931 2/20 0.35
KDR P35968 2/20 0.35
PIK3CA P42336 2/20 0.35
PIK3CB P42338 2/20 0.35
MTOR P42345 2/20 0.35
PIK3CG P48736 2/20 0.35
EPHB4 P54760 2/20 0.35
PRKDC P78527 2/20 0.35
PI4KB Q9UBF8 2/20 0.35
ITK Q08881 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23917564 0.83 FGFR1 (0.43) FGFR1FGFR4FGFR2FGFR3EGFR
SCHEMBL23917271 0.80 BTK (0.40) FGFR1FGFR4FGFR2FGFR3EGFR
SCHEMBL16065725 0.79 PIK3CD (0.53) EGFRPIK3CDABL1HCKSRC
SCHEMBL16665750 0.76 FGFR1 (0.39) FGFR1FGFR4FGFR2FGFR3EGFR
SCHEMBL152637 0.73 PIK3CD (0.49) FGFR1FGFR4FGFR2FGFR3EGFR
SCHEMBL20093476 0.73 VRK1 (0.41) EGFRPIK3CDABL1HCKSRC
SCHEMBL16665792 0.73 SRC (0.45) EGFRPIK3CDSRCPIK3CAPIK3CB
SCHEMBL10855 0.72 MAP4K4 (0.49) MAP4K4PIK3CDPIK3CAPIK3CBMTOR
SCHEMBL23917237 0.71 MAP2K4 (0.57) FGFR1FGFR3EGFRPIK3CDABL1
SCHEMBL16665713 0.71 PIK3CD (0.36) EGFRPIK3CDABL1HCKSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210317140-A1 Heterocyclic Compounds and Methods of Use MEDIVATION TECHNOLOGIES, INC. (US) 2021-10-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210317140-A1 Heterocyclic Compounds and Methods of Use BTK, PIK3CD, PIK3CB FGFR1 2569/4885FGFR4 3243/4885MAP4K4 693/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.