Abiraterone

Abiraterone

SCHEMBL23924960

C[C@]12CC[C@H](O)CC1=CC[C@@H]1[C@@H]2CC[C@]2(C)C(c3cccnc3)=CC[C@@H]12.C[C@]12CC[C@H](O)CC1=CC[C@@H]1[C@@H]2CC[C@]2(C)C(c3cccnc3)=CC[C@@H]12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ARCYP17A1SRD5A1SRD5A2SRD5A3

The experimentally established mechanism targets of Abiraterone. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP17A1 known ✓ P05093 16/20 1.00
AR known ✓ P10275 1/20 0.71
CYP21A2 P08686 6/20 1.00
CYP11B1 P15538 2/20 1.00
CYP3A4 P08684 1/20 1.00
CYP11B2 P19099 1/20 1.00
CDK8 P49336 3/20 0.72
PGR P06401 1/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Abiraterone SCHEMBL16383633 1.00 CYP17A1 (1.00) CYP17A1CYP21A2CYP11B1CYP3A4CYP11B2
Abiraterone SCHEMBL17474701 1.00 CYP17A1 (1.00) CYP17A1CYP21A2CYP11B1CYP3A4CYP11B2
Abiraterone SCHEMBL61108 1.00 CYP17A1 (1.00) CYP17A1CYP21A2CYP11B1CYP3A4CYP11B2
Abiraterone SCHEMBL20459184 1.00 CYP17A1 (1.00) CYP17A1CYP21A2CYP11B1CYP3A4CYP11B2
Abiraterone SCHEMBL8736929 1.00 CYP17A1 (1.00) CYP17A1CYP21A2CYP11B1CYP3A4CYP11B2
Abiraterone SCHEMBL25074918 1.00 CYP17A1 (1.00) CYP17A1CYP21A2CYP11B1CYP3A4CYP11B2
Abiraterone SCHEMBL13272100 1.00 CYP17A1 (1.00) CYP17A1CYP21A2CYP11B1CYP3A4CYP11B2
Abiraterone SCHEMBL19724576 1.00 CYP17A1 (1.00) CYP17A1CYP21A2CYP11B1CYP3A4CYP11B2
Abiraterone SCHEMBL22414103 1.00 CYP17A1 (1.00) CYP17A1CYP21A2CYP11B1CYP3A4CYP11B2
Abiraterone SCHEMBL15700283 1.00 CYP17A1 (1.00) CYP17A1CYP21A2CYP11B1CYP3A4CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4135659-A1 METHODS AND COMPOSITIONS FOR TREATING PROSTATE CANCER Tavanta Therapeutics Hungary Incorporated (HU) 2023-02-22 EP disclosed
WO-2021209945-A1 METHODS AND COMPOSITIONS FOR TREATING PROSTATE CANCER TAVANTA THERAPEUTICS HUNGARY INCORPORATED (HU) 2021-10-21 WO disclosed