SCHEMBL23929026

SCHEMBL23929026

COC(=O)c1ccc(CSc2nccc(O)n2)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.61
SMN1; SMN2 Q16637 5/20 0.55
NPC1 O15118 6/20 0.50
RAB9A P51151 6/20 0.50
MAPT P10636 4/20 0.50
LMNA P02545 3/20 0.50
METAP2 P50579 2/20 0.50
ALDH1A1 P00352 2/20 0.50
PKM P14618 1/20 0.50
MAPK1 P28482 2/20 0.49
POLB P06746 1/20 0.49
TSHR P16473 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
PTGDR2 Q9Y5Y4 1/20 0.47
GSK3A P49840 1/20 0.47
GSK3B P49841 1/20 0.47
CYP1A2 P05177 2/20 0.46
NPSR1 Q6W5P4 1/20 0.46
HPGD P15428 2/20 0.46
CYP3A4 P08684 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28652347 0.86 TP53 (0.60) TP53SMN1; SMN2NPC1RAB9AMAPT
SCHEMBL2302038 0.85 TP53 (0.68) TP53SMN1; SMN2NPC1RAB9AMAPT
SCHEMBL16920966 0.81 NPC1 (0.50) TP53SMN1; SMN2NPC1RAB9AMAPT
SCHEMBL209840 0.80 MAPT (0.61) TP53SMN1; SMN2NPC1MAPTLMNA
SCHEMBL27900976 0.77 METAP2 (0.53) TP53SMN1; SMN2NPC1RAB9AMAPT
SCHEMBL16920960 0.76 HTT (0.51) TP53SMN1; SMN2NPC1RAB9AMAPT
SCHEMBL23962996 0.76 AURKA (0.52) TP53SMN1; SMN2METAP2MAPK1
SCHEMBL16920959 0.75 HSD17B10 (0.65) SMN1; SMN2NPC1RAB9AMAPTMETAP2
SCHEMBL13058926 0.75 NPSR1 (0.47) RAB9AMAPTLMNAMETAP2ALDH1A1
SCHEMBL3919430 0.73 GSK3A (0.62) TP53SMN1; SMN2NPC1RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113549057-B Snail inhibitor and derivative thereof, preparation method, pharmaceutical composition and application 中国药科大学 2023-01-31 CN disclosed
WO-2021213111-A1 SNAIL INHIBITOR, DERIVATIVE THEREOF, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND USE THEREOF 中国药科大学 (CN) 2021-10-28 WO disclosed
WO-2021213111-A1 SNAIL INHIBITOR, DERIVATIVE THEREOF, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND USE THEREOF 中国药科大学 (CN) 2021-10-28 WO disclosed
CN-113549057-A Snail inhibitor and derivative thereof, preparation method, pharmaceutical composition and application 中国药科大学 2021-10-26 CN disclosed