SCHEMBL23934779

SCHEMBL23934779

C#Cc1cccc(Nc2ncnc3cc(C)c(OCCCN4CCOCC4)cc23)c1

nearest known ligand 0.83

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 14/20 0.83
SRC P12931 6/20 0.65
KDR P35968 4/20 0.65
GAK O14976 4/20 0.60
BRAF P15056 3/20 0.60
ERBB2 P04626 3/20 0.60
RIPK2 O43353 3/20 0.60
STK10 O94804 3/20 0.60
PIP4K2C Q8TBX8 3/20 0.60
SLK Q9H2G2 3/20 0.60
BUB1 O43683 2/20 0.60
MAP3K1 Q13233 2/20 0.60
CIT O14578 2/20 0.60
EPHB6 O15197 2/20 0.60
DAPK3 O43293 2/20 0.60
RPS6KA4 O75676 2/20 0.60
STK17B O94768 2/20 0.60
ABCB11 O95342 2/20 0.60
ABL1 P00519 2/20 0.60
LCK P06239 2/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29578659 0.93 EGFR (0.92) EGFRSRCKDRGAKBRAF
SCHEMBL28696278 0.93 EGFR (0.92) EGFRSRCKDRGAKBRAF
SCHEMBL828788 0.91 EGFR (1.00) EGFRSRCKDRGAKBRAF
SCHEMBL29483201 0.91 EGFR (1.00) EGFRSRCKDRGAKBRAF
Hydrochloric Acid SCHEMBL20534441 0.90 EGFR (0.98) EGFRSRCKDRGAKBRAF
Hydrochloric Acid SCHEMBL30133464 0.90 EGFR (0.98) EGFRSRCKDRGAKBRAF
SCHEMBL28700304 0.89 EGFR (0.84) EGFRSRCKDRGAKBRAF
SCHEMBL29579338 0.89 EGFR (0.84) EGFRSRCKDRGAKBRAF
SCHEMBL826406 0.89 EGFR (0.78) EGFRSRCKDRGAKBRAF
SCHEMBL18651673 0.88 EGFR (0.77) EGFRSRCKDRGAKBRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3609875-B1 AN IMPROVED PROCESS FOR THE PREPARATION OF N-(3-ETHYNYLPHENYL)-7-METHOXY-6-(3-MORPHOLINOPROPOXY) QUINAZOLIN -4-AMINE DIHYDROCHLORIDE NATCO PHARMA LTD (IN) 2021-10-20 EP disclosed