SCHEMBL23935201

SCHEMBL23935201

Cn1c(Cc2ccon2)nc2cnc3cccnc3c21

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.36
KDM4E B2RXH2 1/20 0.32
TLR7 Q9NYK1 1/20 0.32
ALDH1A1 P00352 1/20 0.32
USP2 O75604 1/20 0.31
RAB9A P51151 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23922646 0.76 LRRK2 (0.51)
SCHEMBL18658907 0.76 LRRK2 (0.51)
SCHEMBL18606520 0.76 LRRK2 (0.51)
SCHEMBL23934997 0.74 LRRK2 (0.45)
SCHEMBL23934965 0.72 LRRK2 (0.49)
SCHEMBL4302608 0.68 KDM4E (0.40) PDE10AKDM4ETLR7
SCHEMBL4312799 0.66 SMN1; SMN2 (0.40) PDE10ATLR7
SCHEMBL18606425 0.65 JAK1 (0.45)
SCHEMBL27666505 0.65 TLR7 (0.44) TLR7
SCHEMBL12888448 0.65 HPGD (0.42) PDE10ATLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3350178-B1 NOVEL IMIDAZO [4,5-C]QUINOLINE AND IMIDAZO [4,5-C][1,5]NAPHTHYRIDINE DERIVATIVES AS LRRK2 INHIBITORS PFIZER (US) 2021-10-20 EP disclosed