SCHEMBL23937735

SCHEMBL23937735

CC(C)c1nc(NCC2CC2)c2ccccn12

nearest known ligand 0.50

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 20/20 0.50
CYP3A4 P08684 6/20 0.49
CYP2D6 P10635 5/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20673899 0.80 PDE10A (0.41) HTR4CYP3A4
SCHEMBL21958603 0.76 PDE10A (0.39) HTR4CYP3A4CYP2D6
SCHEMBL23937736 0.75 HTR4 (0.42) HTR4CYP3A4CYP2D6
SCHEMBL23937719 0.71 HTR4 (0.42) HTR4CYP3A4CYP2D6
SCHEMBL19699834 0.69 PTPN1 (0.53) HTR4CYP3A4CYP2D6
SCHEMBL21180241 0.69 HTR4 (0.43) HTR4CYP3A4CYP2D6
SCHEMBL20674149 0.69 HTR4 (0.40) HTR4CYP3A4CYP2D6
SCHEMBL20927196 0.68 HTR4 (0.44) HTR4CYP3A4CYP2D6
SCHEMBL28700587 0.67 HTR4 (0.42) HTR4CYP3A4CYP2D6
SCHEMBL23937874 0.67 ACVR1 (0.39) HTR4CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3399968-B1 SELECTIVE INHIBITORS OF CLINICALLY IMPORTANT MUTANTS OF THE EGFR TYROSINE KINASE CS PHARMATECH LTD (KY) 2021-10-20 EP disclosed