SCHEMBL23937771

SCHEMBL23937771

CCn1ncc2ccsc21

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
HASPIN Q8TF76 1/20 0.36
HPGD P15428 1/20 0.35
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
KMT2A Q03164 1/20 0.34
CYP11B2 P19099 1/20 0.33
ADORA1 P30542 4/20 0.32
ADORA3 P0DMS8 2/20 0.32
HTT P42858 1/20 0.32
ADORA2A P29274 2/20 0.31
CYP2C19 P33261 1/20 0.30
RECQL P46063 1/20 0.30
TP53 P04637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3174711 0.74
SCHEMBL16267051 0.72 PLA2G4A (0.37) ALDH1A1KMT2A
SCHEMBL23937806 0.69 HTR2A (0.34) HTR2AHTR2CHPGDALDH1A1KMT2A
SCHEMBL16267053 0.65 ASAH1 (0.41) MEN1ALDH1A1KMT2ACYP2C19
SCHEMBL13217 0.64 RECQL (0.61) MEN1KMT2ARECQL
SCHEMBL21295080 0.63 PDE7A (0.40) HPGDALDH1A1
SCHEMBL21285480 0.61 MAPT (0.40) HTR2AHTR2CHASPINMEN1KMT2A
SCHEMBL23206121 0.61 HTR2C (0.46) HTR2AHTR2CHASPINCYP11B2HTT
SCHEMBL21501930 0.61 HASPIN (0.49) HTR2AHTR2CHASPINHPGDALDH1A1
SCHEMBL18237382 0.61 HASPIN (0.36) HASPINCYP11B2HTTRECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3399968-B1 SELECTIVE INHIBITORS OF CLINICALLY IMPORTANT MUTANTS OF THE EGFR TYROSINE KINASE CS PHARMATECH LTD (KY) 2021-10-20 EP disclosed