SCHEMBL23937773

SCHEMBL23937773

CCc1cnc2c(ccn2C)n1

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BRD9 Q9H8M2 1/20 0.33
APP P05067 1/20 0.33
PDE10A Q9Y233 2/20 0.32
PIK3CB P42338 1/20 0.32
GRM5 P41594 1/20 0.31
DYRK1A Q13627 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17827121 0.84 PIK3CB (0.34) BRD9APPPDE10APIK3CBGRM5
SCHEMBL23937774 0.76 ELANE (0.34)
SCHEMBL16511362 0.76 BRD9 (0.36) BRD9APPPIK3CBGRM5
SCHEMBL13573819 0.74 PIK3CB (0.44) BRD9APPPIK3CBGRM5DYRK1A
SCHEMBL30912393 0.74 MAPK1 (0.39) BRD9APPPIK3CBGRM5
SCHEMBL13573893 0.74 MAPK1 (0.39) BRD9APPPIK3CBGRM5
SCHEMBL20673864 0.74 BRD9 (0.35) BRD9APPPIK3CBGRM5
SCHEMBL12032587 0.70 PIK3CB (0.34) BRD9APPPIK3CBGRM5
SCHEMBL256368 0.70 ELANE (0.42) BRD9PIK3CBGRM5
SCHEMBL17122511 0.70 FGFR3 (0.38) APPPDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3399968-B1 SELECTIVE INHIBITORS OF CLINICALLY IMPORTANT MUTANTS OF THE EGFR TYROSINE KINASE CS PHARMATECH LTD (KY) 2021-10-20 EP disclosed