SCHEMBL23937774

SCHEMBL23937774

CCc1cnc2c(ccn2C2CC2)n1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ELANE P08246 1/20 0.34
CHEK2 O96017 8/20 0.32
CHEK1 O14757 7/20 0.32
CYP11B1 P15538 2/20 0.32
CYP11B2 P19099 2/20 0.32
ALDH1A1 P00352 2/20 0.32
CYP1A2 P05177 2/20 0.32
CASP1 P29466 2/20 0.32
CASP7 P55210 2/20 0.32
HSD17B10 Q99714 2/20 0.32
CLK4 Q9HAZ1 2/20 0.32
CYP2C9 P11712 1/20 0.32
DRD2 P14416 2/20 0.31
SLC6A4 P31645 2/20 0.31
PIP4K2A P48426 1/20 0.31
HTR3A P46098 1/20 0.31
KCNH2 Q12809 1/20 0.31
AURKA O14965 1/20 0.31
INSR P06213 1/20 0.31
CDK1 P06493 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20673865 0.81 CHEK2 (0.35) CHEK2CHEK1CYP11B1CYP11B2ALDH1A1
SCHEMBL21959627 0.76 ELANE (0.33) ELANEAURKAINSRCDK1PDGFRB
SCHEMBL23937773 0.76 BRD9 (0.33)
SCHEMBL21959623 0.73 PDE10A (0.32) CHEK2CHEK1CYP11B1CYP11B2ALDH1A1
SCHEMBL23937881 0.73 PARP1 (0.37) DRD2SLC6A4KCNH2AURKAINSR
SCHEMBL23937732 0.72 CYP11B1 (0.36) CYP11B1CYP11B2DRD2SLC6A4PIP4K2A
SCHEMBL21958686 0.70 DRD2 (0.37) CYP11B1CYP11B2DRD2SLC6A4
SCHEMBL24995507 0.67 PDE10A (0.31)
SCHEMBL23442191 0.65 CHEK2 (0.50) CHEK2CHEK1ALDH1A1CYP1A2CASP1
SCHEMBL16167705 0.65 CNR2 (0.38) ALDH1A1CYP1A2CASP1CASP7HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3399968-B1 SELECTIVE INHIBITORS OF CLINICALLY IMPORTANT MUTANTS OF THE EGFR TYROSINE KINASE CS PHARMATECH LTD (KY) 2021-10-20 EP disclosed