SCHEMBL23938466

SCHEMBL23938466

N/N=C(\NN)c1cc(F)ccc1F

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 3/20 0.47
CES1 P23141 3/20 0.47
CA3 P07451 1/20 0.38
CA6 P23280 1/20 0.38
CA5A P35218 1/20 0.38
CA9 Q16790 1/20 0.38
CA14 Q9ULX7 1/20 0.38
CA5B Q9Y2D0 1/20 0.38
KEAP1 Q14145 1/20 0.35
ALDH1A1 P00352 2/20 0.33
TAS1R3 Q7RTX0 1/20 0.33
TAS1R1 Q7RTX1 1/20 0.33
TAS1R2 Q8TE23 1/20 0.33
MDM2 Q00987 1/20 0.32
ALPL P05186 1/20 0.32
IDO1 P14902 2/20 0.32
GRIN2D O15399 2/20 0.32
GRIN3B O60391 2/20 0.32
GRIN1 Q05586 2/20 0.32
GRIN2A Q12879 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24007285 0.79 CES2 (0.32) CES2CES1KEAP1IDO1
SCHEMBL23938344 0.78 MAP2K2 (0.36) ALDH1A1IDO1GAA
SCHEMBL15489581 0.75 CES2 (0.52) CES2CES1CA3CA6CA5A
SCHEMBL12225512 0.75 CES2 (0.52) CES2CES1CA3CA6CA5A
SCHEMBL801104 0.73 CES2 (0.50) CES2CES1CA3CA6CA5A
SCHEMBL84165 0.73 CES2 (0.50) CES2CES1CA3CA6CA5A
Hydrochloric Acid SCHEMBL7963311 0.73 CES2 (0.50) CES2CES1CA3CA6CA5A
SCHEMBL246382 0.73 CES2 (0.61) CES2CES1KEAP1ALDH1A1TAS1R3
SCHEMBL16359664 0.73 CES2 (0.50) CES2CES1CA3CA6CA5A
SCHEMBL24417687 0.72 CYP11B1 (0.38) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3297438-B1 CCR2 MODULATORS CHEMOCENTRYX INC (US) 2021-10-20 EP disclosed