SCHEMBL2394573

SCHEMBL2394573

N[C@@H](COc1cccnc1)c1ccccc1

nearest known ligand 0.69

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SCN4A P35499 7/20 0.69
AKT1 P31749 3/20 0.57
CHRNB2 P17787 4/20 0.45
CHRNA4 P43681 4/20 0.45
CFTR P13569 1/20 0.44
SLC6A2 P23975 1/20 0.44
SLC6A4 P31645 1/20 0.44
SLC6A3 Q01959 1/20 0.44
GOPC Q9HD26 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19686108 1.00 SCN4A (0.69) SCN4AAKT1CHRNB2CHRNA4CFTR
SCHEMBL4345367 0.82 SCN4A (1.00) SCN4A
SCHEMBL12847267 0.82 SCN4A (1.00) SCN4A
SCHEMBL19686196 0.81 SCN4A (0.76) SCN4AAKT1SLC6A2SLC6A4SLC6A3
SCHEMBL19686206 0.79 SCN4A (0.62) SCN4AAKT1
SCHEMBL19686194 0.77 SCN4A (0.58) SCN4AAKT1
SCHEMBL23406075 0.76 SCN4A (0.57) SCN4AAKT1
SCHEMBL29743841 0.76 SCN4A (0.57) SCN4AAKT1
SCHEMBL23406078 0.76 SCN4A (0.57) SCN4AAKT1
SCHEMBL27674373 0.75 CHRNB2 (0.50) AKT1CHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8012901-B1 Method of synthesizing enantiopure mexiletine analogues and novel β-thiophenoxy and pyridyl ethers NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2011-09-06 US disclosed
US-8012901-B1 Method of synthesizing enantiopure mexiletine analogues and novel β-thiophenoxy and pyridyl ethers NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2011-09-06 US disclosed
US-8012901-B1 Method of synthesizing enantiopure mexiletine analogues and novel β-thiophenoxy and pyridyl ethers NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2011-09-06 US disclosed