SCHEMBL2394601

SCHEMBL2394601

Cc1ccccc1OC/C(=N\O)c1ccc(Cl)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.61
MEN1 O00255 3/20 0.50
KMT2A Q03164 3/20 0.50
CYP1A2 P05177 1/20 0.50
CYP2C19 P33261 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
SLC6A4 P31645 1/20 0.48
MAPT P10636 5/20 0.44
POLB P06746 1/20 0.43
ALDH1A1 P00352 1/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
RXRA P19793 1/20 0.42
RXRB P28702 1/20 0.42
RXRG P48443 1/20 0.42
NOTUM Q6P988 1/20 0.42
AOC2 O75106 1/20 0.42
MAOA P21397 1/20 0.42
MAOB P27338 1/20 0.42
HTT P42858 1/20 0.42
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2394607 1.00 GAA (0.61) GAAMEN1KMT2ACYP1A2CYP2C19
SCHEMBL2396381 0.87 GAA (0.63) GAAMEN1KMT2ASLC6A4MAPT
SCHEMBL2396384 0.87 GAA (0.63) GAAMEN1KMT2ASLC6A4MAPT
SCHEMBL2395009 0.86 L3MBTL1 (0.56) GAAMEN1KMT2ATDP1SLC6A4
SCHEMBL2395015 0.86 L3MBTL1 (0.56) GAAMEN1KMT2ATDP1SLC6A4
SCHEMBL2394584 0.83 GAA (0.48) GAAMEN1KMT2ACYP1A2SLC6A4
SCHEMBL2394591 0.83 GAA (0.48) GAAMEN1KMT2ACYP1A2SLC6A4
SCHEMBL2395102 0.80 MAPT (0.65) MEN1KMT2ACYP1A2CYP2C19TDP1
SCHEMBL2396595 0.80 TDP1 (0.49) GAAMEN1KMT2ACYP1A2CYP2C19
SCHEMBL2396592 0.80 TDP1 (0.49) GAAMEN1KMT2ACYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8012901-B1 Method of synthesizing enantiopure mexiletine analogues and novel β-thiophenoxy and pyridyl ethers NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2011-09-06 US disclosed