SCHEMBL23950289

SCHEMBL23950289

CSCCn1cnc2c(-c3cccnc3)nc(-c3ccc(Cl)cc3)cc2c1=O

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 3/20 0.40
ADORA2A P29274 2/20 0.40
GRM2 Q14416 2/20 0.39
PSD A5PKW4 3/20 0.38
CYP2C9 P11712 4/20 0.37
CYP2C19 P33261 4/20 0.37
CYP3A4 P08684 3/20 0.37
CYP1A2 P05177 2/20 0.37
GAA P10253 1/20 0.37
CYP2E1 P05181 2/20 0.36
CYP2A6 P11509 2/20 0.36
CYP2B6 P20813 2/20 0.36
CYP19A1 P11511 1/20 0.35
MAPT P10636 1/20 0.35
PSMB2 P49721 1/20 0.35
DHPS P49366 1/20 0.35
KDM4E B2RXH2 1/20 0.35
POLB P06746 1/20 0.35
CNR1 P21554 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23950296 0.89 GRM2 (0.38) ADORA1ADORA2AGRM2CYP2C9CYP2C19
SCHEMBL26287834 0.88 ADORA2A (0.39) ADORA1ADORA2AGRM2PSDCYP2C9
SCHEMBL23925606 0.87 PSD (0.40) ADORA1ADORA2AGRM2PSDCYP2C9
SCHEMBL23951143 0.86 SYK (0.45)
SCHEMBL23950718 0.85 PSD (0.43) ADORA1ADORA2AGRM2PSDCYP2C9
SCHEMBL23390267 0.84 PSD (0.41) ADORA1ADORA2AGRM2PSDCYP2C9
SCHEMBL23416773 0.84 CYP3A4 (0.39) ADORA1ADORA2AGRM2PSDCYP2C9
SCHEMBL23925559 0.81 PSD (0.38) ADORA1ADORA2AGRM2PSDCYP2C9
SCHEMBL26290323 0.80 CYP2A6 (0.49) ADORA1ADORA2AGRM2CYP2C9CYP2C19
SCHEMBL30102059 0.80 PIM1 (0.39) ADORA1ADORA2AGRM2PSDCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021210970-A1 PYRIDOPYRIMIDINONE DERIVATIVES AND THEIR USE AS ARYL HYDROCARBON RECEPTOR MODULATORS DONG-A ST CO., LTD. (KR) 2021-10-21 WO disclosed