SCHEMBL23950296

SCHEMBL23950296

CSCCn1cnc2c(-c3cccnc3)nc(-c3ccc(C(F)(F)F)cc3)cc2c1=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 1/20 0.38
PIM1 P11309 2/20 0.37
PTGS1 P23219 1/20 0.36
PTGS2 P35354 1/20 0.36
ADORA2A P29274 2/20 0.36
ADORA1 P30542 2/20 0.36
TOP1 P11387 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
EGLN1 Q9GZT9 1/20 0.35
S1PR1 P21453 1/20 0.35
NPY5R Q15761 1/20 0.35
MET P08581 1/20 0.35
CYP2E1 P05181 1/20 0.34
CYP2A6 P11509 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2B6 P20813 1/20 0.34
CYP2C19 P33261 1/20 0.34
NPC1 O15118 1/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23950289 0.89 ADORA1 (0.40) GRM2ADORA2AADORA1CYP2E1CYP2A6
SCHEMBL23950293 0.88 PTGS2 (0.42) GRM2PIM1PTGS1PTGS2ADORA2A
SCHEMBL23950265 0.87 EGLN1 (0.39) GRM2PIM1PTGS1PTGS2TOP1
SCHEMBL23950531 0.85 PIM1 (0.41) PIM1PTGS1PTGS2TOP1SMN1; SMN2
SCHEMBL23390502 0.85 SMN1; SMN2 (0.38) GRM2PIM1PTGS1PTGS2ADORA2A
SCHEMBL23951143 0.83 SYK (0.45) PIM1
SCHEMBL30102064 0.83 PIM1 (0.37) GRM2PIM1PTGS1PTGS2ADORA2A
SCHEMBL23951123 0.83 PIM1 (0.37) GRM2PIM1PTGS1PTGS2ADORA2A
SCHEMBL23950264 0.82 EGLN1 (0.38) GRM2PIM1PTGS1PTGS2ADORA2A
SCHEMBL23950768 0.82 EGLN1 (0.38) GRM2PIM1PTGS1PTGS2ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021210970-A1 PYRIDOPYRIMIDINONE DERIVATIVES AND THEIR USE AS ARYL HYDROCARBON RECEPTOR MODULATORS DONG-A ST CO., LTD. (KR) 2021-10-21 WO disclosed