SCHEMBL23950392

SCHEMBL23950392

CC(C)c1nn(CC(=O)N[C@H]2CCC(=O)N(CC3CC3)C2)c(=O)c2cc(C3CC3)nn12

nearest known ligand 0.57

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 11/20 0.57
KCNH2 Q12809 1/20 0.40
THRB P10828 2/20 0.36
SLC18A2 Q05940 1/20 0.34
TP53 P04637 2/20 0.34
CHRNA7 P36544 2/20 0.33
CHRNA1 P02708 1/20 0.33
CHRNA3 P32297 1/20 0.33
HTR3A P46098 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23950390 1.00 NLRP3 (0.57) NLRP3KCNH2THRBSLC18A2TP53
SCHEMBL23950388 1.00 NLRP3 (0.57) NLRP3KCNH2THRBSLC18A2TP53
SCHEMBL25752826 0.89 NLRP3 (0.61) NLRP3KCNH2THRBSLC18A2TP53
SCHEMBL23950816 0.89 NLRP3 (0.61) NLRP3KCNH2THRBSLC18A2TP53
SCHEMBL23950811 0.89 NLRP3 (0.61) NLRP3KCNH2THRBSLC18A2TP53
SCHEMBL25753229 0.81 NLRP3 (0.56) NLRP3KCNH2THRBSLC18A2TP53
SCHEMBL23950385 0.80 NLRP3 (0.61) NLRP3KCNH2THRBTP53CHRNA7
SCHEMBL23950511 0.79 NLRP3 (0.62) NLRP3KCNH2THRBTP53
SCHEMBL23925343 0.79 NLRP3 (0.62) NLRP3KCNH2THRBSLC18A2
SCHEMBL23925344 0.79 NLRP3 (0.62) NLRP3KCNH2THRBSLC18A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021209552-A1 PYRAZOLO[1,5-D][1,2,4]TRIAZINE-5(4H)-ACETAMIDES AS INHIBITORS OF THE NLRP3 INFLAMMASOME PATHWAY JANSSEN PHARMACEUTICA NV (BE) 2021-10-21 WO disclosed