SCHEMBL23950631

SCHEMBL23950631

CC(C)c1nn(CC(=O)N/C(N)=C/C=C(\N)C(F)(F)F)c(=O)c2cc(C3CC3)nn12

nearest known ligand 0.53

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 13/20 0.53
GPR139 Q6DWJ6 2/20 0.35
KCNH2 Q12809 1/20 0.35
THRB P10828 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23950801 0.80 NLRP3 (0.58) NLRP3GPR139KCNH2THRB
SCHEMBL23950172 0.78 NLRP3 (0.60) NLRP3GPR139KCNH2THRB
SCHEMBL23950511 0.77 NLRP3 (0.62) NLRP3KCNH2THRB
SCHEMBL23950466 0.76 NLRP3 (0.59) NLRP3GPR139KCNH2
SCHEMBL25242095 0.76 NLRP3 (0.64) NLRP3GPR139KCNH2THRB
SCHEMBL30040964 0.76 NLRP3 (0.53) NLRP3GPR139KCNH2
SCHEMBL23950385 0.75 NLRP3 (0.61) NLRP3KCNH2THRB
SCHEMBL25283591 0.75 NLRP3 (0.58) NLRP3KCNH2THRB
SCHEMBL23950219 0.75 NLRP3 (0.58) NLRP3KCNH2THRB
SCHEMBL23950360 0.75 NLRP3 (0.58) NLRP3KCNH2THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021209552-A1 PYRAZOLO[1,5-D][1,2,4]TRIAZINE-5(4H)-ACETAMIDES AS INHIBITORS OF THE NLRP3 INFLAMMASOME PATHWAY JANSSEN PHARMACEUTICA NV (BE) 2021-10-21 WO disclosed