SCHEMBL23950972

SCHEMBL23950972

O=c1c2cc(-c3cnc(C(F)(F)F)nc3)nc(-c3cccnc3)c2ncn1C1CCC(O)C1

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CLK1 P49759 1/20 0.37
DYRK1A Q13627 1/20 0.37
KCNH2 Q12809 1/20 0.36
PIM1 P11309 13/20 0.34
HTR2B P41595 1/20 0.33
HTR6 P50406 1/20 0.33
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
ABL1 P00519 1/20 0.32
MAP4K1 Q92918 1/20 0.32
HSP90AA1 P07900 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23950974 1.00 CLK1 (0.37) CLK1DYRK1AKCNH2PIM1HTR2B
SCHEMBL23925639 0.91 CLK1 (0.36) CLK1DYRK1AKCNH2PIM1HSP90AA1
SCHEMBL23950604 0.91 CLK1 (0.36) CLK1DYRK1AKCNH2PIM1HSP90AA1
SCHEMBL23951140 0.90 CYP11B1 (0.39) CLK1DYRK1AKCNH2PIM1HTR2B
SCHEMBL23925575 0.90 CYP11B1 (0.39) CLK1DYRK1AKCNH2PIM1HTR2B
SCHEMBL23925713 0.90 CYP11B1 (0.39) CLK1DYRK1AKCNH2PIM1HTR2B
SCHEMBL23925582 0.87 CYP2A6 (0.39) CLK1DYRK1AKCNH2PIM1
SCHEMBL30101964 0.87 CYP2A6 (0.39) CLK1DYRK1AKCNH2PIM1
SCHEMBL23950769 0.87 CYP2A6 (0.39) CLK1DYRK1AKCNH2PIM1
SCHEMBL25463141 0.86 CLK1 (0.38) CLK1DYRK1AKCNH2PIM1CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021210970-A1 PYRIDOPYRIMIDINONE DERIVATIVES AND THEIR USE AS ARYL HYDROCARBON RECEPTOR MODULATORS DONG-A ST CO., LTD. (KR) 2021-10-21 WO disclosed